Global Patent Index - EP 0000032 B1

EP 0000032 B1 19820519 - DI- AND TRI-SUBSTITUTED THIAZOLES, THEIR PREPARATION, THEIR USE IN PHARMACEUTICALS AND INTERMEDIATE COMPOUNDS

Title (en)

DI- AND TRI-SUBSTITUTED THIAZOLES, THEIR PREPARATION, THEIR USE IN PHARMACEUTICALS AND INTERMEDIATE COMPOUNDS

Publication

EP 0000032 B1 19820519 (EN)

Application

EP 78100053 A 19780601

Priority

  • US 80240377 A 19770601
  • US 89707578 A 19780417

Abstract (en)

[origin: US4260609A] Di- and tri- substituted thiazoles, one substituent being a 3-amino-2-OR-propoxy group are disclosed. The thiazoles have beta -adrenergic blocking activity.

IPC 1-7

C07D 277/34; C07D 277/36; C07D 277/56; C07D 401/04; C07D 417/12; C07D 263/06; A61K 31/44; A61K 31/425; A61K 31/535; A61K 31/495

IPC 8 full level

A61K 31/425 (2006.01); A61K 31/426 (2006.01); A61K 31/44 (2006.01); A61K 31/505 (2006.01); A61K 31/535 (2006.01); A61P 25/02 (2006.01); C07D 263/06 (2006.01); C07D 277/20 (2006.01); C07D 277/34 (2006.01); C07D 277/36 (2006.01); C07D 277/56 (2006.01); C07D 417/04 (2006.01); C07D 417/06 (2006.01); C07D 417/12 (2006.01)

CPC (source: EP US)

A61K 31/425 (2013.01 - EP US); A61K 31/44 (2013.01 - EP US); A61K 31/505 (2013.01 - EP US); A61K 31/535 (2013.01 - EP US); A61P 25/02 (2017.12 - EP); C07D 263/06 (2013.01 - EP US); C07D 277/34 (2013.01 - EP US); C07D 277/36 (2013.01 - EP US); C07D 277/56 (2013.01 - EP US); C07D 417/04 (2013.01 - EP US); C07D 417/12 (2013.01 - EP US)

Designated contracting state (EPC)

BE CH DE FR GB LU NL SE

DOCDB simple family (publication)

US 4260609 A 19810407; EP 0000032 A1 19781220; EP 0000032 B1 19820519; JP S543063 A 19790111; JP S631308 B2 19880112

DOCDB simple family (application)

US 89707578 A 19780417; EP 78100053 A 19780601; JP 6501878 A 19780601