Global Patent Index - EP 0000889 A1

EP 0000889 A1 19790307 - 3"-N-Demethyl-3"-N-substituted-4,6-di-0-(aminoglycosyl)-1,3-diaminocyclitols, methods for their preparation and their application as antibiotics.

Title (en)

3"-N-Demethyl-3"-N-substituted-4,6-di-0-(aminoglycosyl)-1,3-diaminocyclitols, methods for their preparation and their application as antibiotics.

Title (de)

3"-N-Demethyl-3"-N-substituierte-4,6-di-0-(Aminoglycosyl)-1,3-Diaminocyclitole, Verfahren zu deren Herstellung und deren Verwendung als Antibiotika.

Title (fr)

3"-N-Démethyl-3"-N-substitué-4,6-di-0-(aminoglycosyl)-1,3-diaminocyclitols, méthodes pour leur préparation et leur application comme antibiotiques.

Publication

EP 0000889 A1 19790307 (DE)

Application

EP 78100601 A 19780807

Priority

DE 2737264 A 19770818

Abstract (en)

[origin: ES472640A1] The invention includes, as novel compounds, aminoglycoside antibiotics of the 4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols which are 3-N''-substituted. Also included in the invention are compositions containing said novel compounds and methods for the use of said compounds and compositions.

Abstract (de)

Pseudotrisaccharide der Formel <IMAGE> in der X für einen Rest <IMAGE> steht, und Y einen Rest <IMAGE> bezeichnet, U, V, W Wasserstoff oder Hydroxy bedeuten, Z Wasserstoff, Hydroxy oder Amino sein kann und R für Alkyl (ausser Methyl), Alkenyl, Alkinyl, Cycloalkyl, Cycloalkenyl, Cycloalkyl-alkyl, Cycloalkenylalkyl, Aryl oder Aralkyl steht, sind antimikrobielle Mittel mit einem breiten Wirkungsspektrum und besonderer Wirksamkeit gegen gramnegative Bakterien.

IPC 1-7

C07H 15/22; A61K 31/70

IPC 8 full level

A61K 31/70 (2006.01); A61K 31/7028 (2006.01); A61K 31/7034 (2006.01); A61K 31/7036 (2006.01); A61P 31/04 (2006.01); C07H 15/22 (2006.01); C07H 15/234 (2006.01); C07H 15/236 (2006.01)

CPC (source: EP US)

A61P 31/04 (2018.01 - EP); C07H 15/234 (2013.01 - EP US)

Citation (search report)

Designated contracting state (EPC)

BE CH DE FR GB NL

DOCDB simple family (publication)

EP 0000889 A1 19790307; EP 0000889 B1 19810429; AR 220145 A1 19801015; AT 367431 B 19820712; AT A601878 A 19811115; AU 3901478 A 19800221; AU 519849 B2 19811224; DE 2737264 A1 19790301; DE 2860651 D1 19810806; ES 472640 A1 19790216; IE 47429 B1 19840321; IE 781659 L 19790218; IT 1112698 B 19860120; IT 7826782 A0 19780816; JP S5441847 A 19790403; NZ 188147 A 19800428; US 4224315 A 19800923; ZA 784683 B 19790829

DOCDB simple family (application)

EP 78100601 A 19780807; AR 27335078 A 19780818; AT 601878 A 19780818; AU 3901478 A 19780817; DE 2737264 A 19770818; DE 2860651 T 19780807; ES 472640 A 19780817; IE 165978 A 19780817; IT 2678278 A 19780816; JP 9915878 A 19780816; NZ 18814778 A 19780815; US 93170878 A 19780807; ZA 784683 A 19780817