Global Patent Index - EP 0047323 A1

EP 0047323 A1 19820317 - 1,4-NAPHTHOQUINONE DERIVATIVES AND USE THEREOF.

Title (en)

1,4-NAPHTHOQUINONE DERIVATIVES AND USE THEREOF.

Title (de)

1,4-NAPHTHOCHINONDERIVATE UND DEREN VERWENDUNG.

Title (fr)

DERIVES DE 1,4-NAPHTHOQUINONE ET LEUR UTILISATION.

Publication

EP 0047323 A1 19820317 (EN)

Application

EP 81900552 A 19810306

Priority

JP 2967580 A 19800306

Abstract (en)

[origin: WO8102574A1] 1, 4-naphthoquinone derivatives represented by the following general formula: (FORMULA) (wherein R1 represents a hydrogen atom, a hydroxy group, a lower alkoxy group or an arylthio group, R2 represents a carboxy group, an esterified carboxy group or an amidated carboxy group or, when taken together, R1 and R2 form a group of -0- (FORMULA) C-, R3 represents a hydrogen atom or a lower alkyl group, R4 represents a lower alkyl group, R5 represents a hydrogen atom or a halogen atom, and R6 represents a hydrogen atom, a lower alkyl group or a lower alkanoyl group), and the salts of the carboxy group thereof, which are novel compounds having an anti-coccidium activity, and which can be obtained by synthesis or, partly, by cultivation of Streptomyces auranticolor.

Abstract (fr)

Des derives de 1, 4-naphthoquinone sont representes par la formule generale suivante: (FORMULE) (ou R1 represente un atome d'hydrogene, un groupe hydroxy, un groupe alkoxy inferieur ou un groupe arylthio, R2 represente un groupe carboxy, un groupe carboxy esterifie ou un groupe carboxy amide lorsqu'ils sont pris ensemble, R1 et R2 forment un groupe de -O-C-, R3 represente un atome d'hydrogene (FORMULE) ou un groupe alkyl inferieur, R4 represente un groupe alkyle inferieur, R5 represente un atome d'hydrogene ou un atome d'halogene, et R6 represente un atome d'hydrogene, un groupe alkyle inferieur ou un groupe alcanoyle inferieur), et les sels de leur groupe carboxy, qui sont des nouveaux composes ayant une activite anti-coccidium, et qui peuvent etre obtenus par synthese ou, partiellement, par culture de Streptomyces auranticolor.

IPC 1-7

C07C 65/00; C07C 69/94; C07C 103/22; C07C 103/76; C07C 103/84; C07C 149/40; C07D 311/78; C12P 7/26; C12P 17/06

IPC 8 full level

A61K 31/12 (2006.01); A61K 31/16 (2006.01); A61K 31/165 (2006.01); A61K 31/19 (2006.01); A61K 31/215 (2006.01); A61K 31/22 (2006.01); A61K 31/35 (2006.01); A61K 31/352 (2006.01); A61K 31/365 (2006.01); A61K 31/66 (2006.01); A61P 33/02 (2006.01); C07C 50/10 (2006.01); C07C 65/00 (2006.01); C07C 65/03 (2006.01); C07C 65/105 (2006.01); C07C 66/00 (2006.01); C07C 67/00 (2006.01); C07C 69/02 (2006.01); C07C 69/94 (2006.01); C07C 69/95 (2006.01); C07C 231/00 (2006.01); C07C 233/12 (2006.01); C07C 235/46 (2006.01); C07C 235/84 (2006.01); C07C 275/54 (2006.01); C07C 313/00 (2006.01); C07C 323/22 (2006.01); C07C 323/61 (2006.01); C07D 311/78 (2006.01); C07F 9/38 (2006.01); C07F 9/40 (2006.01); C12P 7/40 (2006.01); C12P 7/66 (2006.01); C12P 17/06 (2006.01); C12R 1/465 (2006.01)

CPC (source: EP US)

A61P 33/02 (2017.12 - EP); C07C 66/00 (2013.01 - EP US); C07C 323/00 (2013.01 - EP US); C07D 311/78 (2013.01 - EP US); C12P 7/40 (2013.01 - EP US); C12P 17/06 (2013.01 - EP US)

Designated contracting state (EPC)

AT CH DE FR GB LU NL SE

DOCDB simple family (publication)

EP 0047323 A1 19820317; EP 0047323 A4 19820713; EP 0047323 B1 19841010; AT E9790 T1 19841015; JP H0115491 B2 19890317; JP S56125335 A 19811001; US 4414226 A 19831108; US 4530845 A 19850723; WO 8102574 A1 19810917

DOCDB simple family (application)

EP 81900552 A 19810306; AT 81900552 T 19810306; JP 2967580 A 19800306; JP 8100046 W 19810306; US 31789781 A 19811030; US 51126883 A 19830706