Global Patent Index - EP 0069377 A2

EP 0069377 A2 19830112 - Antibacterial penem derivatives.

Title (en)

Antibacterial penem derivatives.

Title (de)

Antibakterielle Penemderivate.

Title (fr)

Dérivés de pénème antibactériens.

Publication

EP 0069377 A2 19830112 (EN)

Application

EP 82105989 A 19820705

Priority

  • GB 8121108 A 19810708
  • GB 8207136 A 19820311

Abstract (en)

Penem derivative of the formula I <CHEM> in which R is hydrogen or a carboxyl esterifying group, R<1> is phenyl, napthyl, thienyl, pyridyl, quinolyl or isoquinolyl being unsubstituted or substituted by one, two or three of the same or different substituents selected from halogen, hydroxy, amino, nitro, cyano, azido, alkyl, alkoxy, alkanesulfenyl, alkanesulfinyl, alkanesulfonyl, alkanoyl, alkoxycarbonyl, alkanoyloxy, carbamoyl, ureido, carbamoyloxy, alkanoylamino, aminosulfamoyl, sulfamoyl, guanidino, trifluormethyl, trifluormethanesulfenyl, trifluormethanesulfinyl, trifluormethanesulfonoyl and formyl, which may be substituted by one, two or three lower alkyl groups being the same or different. R<2> represents a hydrogen atom or a optionally protected hydroxyl group, or a salt thereof, process for the production thereof and antibacterial pharmaceutical preparations comprising them.

IPC 1-7

C07D 499/00; C07D 205/08; A61K 31/43

IPC 8 full level

C07D 499/00 (2006.01); C07D 205/08 (2006.01); C07D 205/09 (2006.01); C07D 333/38 (2006.01); C07D 499/88 (2006.01); C07F 7/18 (2006.01)

CPC (source: EP KR US)

C07D 205/08 (2013.01 - EP US); C07D 205/09 (2013.01 - EP US); C07D 333/38 (2013.01 - EP US); C07D 499/00 (2013.01 - KR); C07D 499/88 (2013.01 - EP US); C07F 7/1804 (2013.01 - EP US)

Designated contracting state (EPC)

AT BE CH DE FR GB IT LI LU NL SE

DOCDB simple family (publication)

EP 0069377 A2 19830112; EP 0069377 A3 19830413; EP 0069377 B1 19880622; AU 562008 B2 19870528; AU 7097287 A 19870827; AU 7097387 A 19870827; AU 7097487 A 19870827; AU 8570282 A 19830113; CA 1225392 A 19870811; DE 3278689 D1 19880728; ES 513672 A0 19830401; ES 516863 A0 19840116; ES 516864 A0 19830916; ES 8305366 A1 19830401; ES 8308567 A1 19830916; ES 8402309 A1 19840116; FI 77661 B 19881230; FI 77661 C 19890410; FI 822401 A0 19820706; FI 822401 L 19830109; GB 2102798 A 19830209; GB 2102798 B 19851211; GB 2151630 A 19850724; GB 2151630 B 19860212; GB 8500841 D0 19850220; GR 75500 B 19840724; IE 54585 B1 19891206; IE 821641 L 19830108; IL 66245 A0 19821130; IL 66245 A 19880531; KR 840000557 A 19840225; KR 890001885 B1 19890529; PT 75197 A 19820801; PT 75197 B 19850107; US 4585767 A 19860429; US 4772692 A 19880920

DOCDB simple family (application)

EP 82105989 A 19820705; AU 7097287 A 19870402; AU 7097387 A 19870402; AU 7097487 A 19870402; AU 8570282 A 19820707; CA 406827 A 19820707; DE 3278689 T 19820705; ES 513672 A 19820702; ES 516863 A 19821027; ES 516864 A 19821027; FI 822401 A 19820706; GB 8219773 A 19820708; GB 8500841 A 19850114; GR 820168652 A 19820706; IE 164182 A 19820707; IL 6624582 A 19820706; KR 820003013 A 19820706; PT 7519782 A 19820706; US 61970384 A 19840614; US 85499886 A 19860422