Global Patent Index - EP 0154417 A2

EP 0154417 A2 19850911 - 7-Amino-3-substituted-methyl-3-cephem-4-carboxylic acid and lower alkylsilyl derivatives thereof, and their production.

Title (en)

7-Amino-3-substituted-methyl-3-cephem-4-carboxylic acid and lower alkylsilyl derivatives thereof, and their production.

Title (de)

7-Amino-3-substituierte Methyl-3-Cephem-4-carboxylsäure und seine niedrigen Alkylsilyl-Derivate und seine Herstellung.

Title (fr)

Acide 7-amino-3-méthyl substitué-3-céphem-4-carboxylique et ses dérivés alkyl inférieur silyl, et sa préparation.

Publication

EP 0154417 A2 19850911 (EN)

Application

EP 85300823 A 19850207

Priority

JP 2411084 A 19840210

Abstract (en)

Various 7-amino-3-substituted-methyl-3-cephem-4-carboxylic acids and lower alkylsilyl derivatives such as 7-amino-3-(2,3-cyclopenteno-1-pyridiniomethyl)-3-cephem-4-carboxylic acid iodide and trimethylsilyl 7-trimethyl- silylamino-3-(5,6,7,8-tetrahydro-2-isoquinoliniomethyl)-3-cephem-4-carboxylate iodide are valuable intermediates in the preparation of cephalosporin antibacterial agents. A new process for the preparation of these acids and derivatives has been devised.

IPC 1-7

C07D 501/18

IPC 8 full level

C07D 501/04 (2006.01); A61K 31/545 (2006.01); C07D 215/06 (2006.01); C07D 231/06 (2006.01); C07D 501/16 (2006.01); C07D 501/18 (2006.01); C07D 501/20 (2006.01); C07D 501/38 (2006.01); C07D 501/46 (2006.01); C07D 501/58 (2006.01)

CPC (source: EP KR US)

C07D 501/18 (2013.01 - EP US); C07D 501/38 (2013.01 - KR); Y02P 20/55 (2015.11 - EP US)

Designated contracting state (EPC)

DE FR GB IT

DOCDB simple family (publication)

EP 0154417 A2 19850911; EP 0154417 A3 19860611; ES 540200 A0 19861116; ES 554060 A0 19871101; ES 8700861 A1 19861116; ES 8800241 A1 19871101; JP S60169486 A 19850902; KR 850005845 A 19850926; KR 920002869 B1 19920406; US 4699980 A 19871013; US 4845211 A 19890704

DOCDB simple family (application)

EP 85300823 A 19850207; ES 540200 A 19850207; ES 554060 A 19860416; JP 2411084 A 19840210; KR 850000823 A 19850209; US 4666187 A 19870504; US 69958485 A 19850208