EP 0179855 B1 19920729 - DOPAMINE AGONISTS
Title (en)
DOPAMINE AGONISTS
Publication
Application
Priority
US 60000884 A 19840413
Abstract (en)
[origin: US4540691A] Compounds are disclosed having the formula: <IMAGE> wherein: R1 is H, OH, -OCH3, -CH2OH, -NH2, -NHMe, -NHEt, -NMe2, -NEt2, <IMAGE> R2 is H, -CH3, or <IMAGE> R3 is phenyl, benzyl, or 1-4 carbon alkyl; R4 is H, -CH3, -CH2OH, -CH2-CN, -CH2-S-Me, CH2-S-CN, or <IMAGE> R5 is H, 1-4 carbon alkyl, alkenyl, or alkynyl, or aralkyl having a 1-4 carbon alkylene moiety; and A is -CH2-or -CH2CH2-, and pharmaceutically-acceptable salts thereof. Pharmaceutical preparations using these compounds and a method for inducing a dopaminergic response by administering these compounds are also disclosed.
IPC 1-7
A61K 31/535; A61K 31/55; C07D 265/36; C07D 267/14; C07D 413/02
IPC 8 full level
A61K 31/535 (2006.01); A61K 31/55 (2006.01); C07D 265/00 (2006.01); C07D 265/34 (2006.01); C07D 265/36 (2006.01); C07D 267/00 (2006.01); C07D 267/12 (2006.01); C07D 267/14 (2006.01); C07D 409/00 (2006.01); C07D 413/02 (2006.01); C07D 413/06 (2006.01)
CPC (source: EP US)
C07D 265/34 (2013.01 - EP US); C07D 267/12 (2013.01 - EP US); C07D 413/06 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE CH DE FR GB IT LI LU NL SE
DOCDB simple family (publication)
US 4540691 A 19850910; AT E78688 T1 19920815; AU 4233985 A 19851101; AU 580597 B2 19890119; CA 1264741 A 19900123; DE 3586411 D1 19920903; DE 3586411 T2 19930107; EP 0179855 A1 19860507; EP 0179855 A4 19860821; EP 0179855 B1 19920729; ES 542229 A0 19870716; ES 557024 A0 19871216; ES 8707207 A1 19870716; ES 8801228 A1 19871216; IE 58384 B1 19930908; IE 850939 L 19851013; JP S61501854 A 19860828; WO 8504582 A1 19851024; ZA 852704 B 19851224
DOCDB simple family (application)
US 60000884 A 19840413; AT 85902262 T 19850410; AU 4233985 A 19850410; CA 478967 A 19850412; DE 3586411 T 19850410; EP 85902262 A 19850410; ES 542229 A 19850412; ES 557024 A 19860814; IE 93985 A 19850412; JP 50186885 A 19850410; US 8500644 W 19850410; ZA 852704 A 19850411