Global Patent Index - EP 0417059 A3

EP 0417059 A3 19910502 - BICYCLIC TETRAHYDROXYLATED PYRROLIZIDINES

Title (en)

BICYCLIC TETRAHYDROXYLATED PYRROLIZIDINES

Publication

EP 0417059 A3 19910502 (EN)

Application

EP 90870138 A 19900904

Priority

US 40480089 A 19890908

Abstract (en)

[origin: EP0417059A2] Novel bicyclic tetrahydroxylated pyrrolizidines are disclosed which are inhibitors of glycosidase enzymes. A preferred inhibitor is 1 alpha ,2 alpha ,6 alpha ,7 alpha ,7 alpha beta -1,2,6-7-tetrahydroxypyrrolizidine. It is synthesized from D-glycero-D-gulo-heptono-1,4-lactone.

IPC 1-7

C07D 487/04; C07F 7/18; C07D 491/22; A61K 31/40

IPC 8 full level

C07D 487/04 (2006.01); A61K 31/40 (2006.01); A61P 3/08 (2006.01); C07D 317/10 (2006.01); C07D 491/04 (2006.01); C07D 491/22 (2006.01); C07D 493/04 (2006.01)

CPC (source: EP US)

A61P 3/08 (2017.12 - EP); C07D 317/10 (2013.01 - EP US); C07D 491/04 (2013.01 - EP US); C07D 493/04 (2013.01 - EP US)

Citation (search report)

EP 0328508 A2 19890816 - SEARLE & CO [US]

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB GR IT LI LU NL SE

DOCDB simple family (publication)

EP 0417059 A2 19910313; EP 0417059 A3 19910502; CA 2024840 A1 19910309; JP H03106883 A 19910507; US 4992460 A 19910212

DOCDB simple family (application)

EP 90870138 A 19900904; CA 2024840 A 19900907; JP 23886290 A 19900907; US 40480089 A 19890908