Global Patent Index - EP 0538374 A4

EP 0538374 A4 19930519 - ASPARTIC PROTEASE INHIBITORS

Title (en)

ASPARTIC PROTEASE INHIBITORS

Publication

EP 0538374 A4 19930519 (EN)

Application

EP 91913442 A 19910703

Priority

US 54946090 A 19900706

Abstract (en)

[origin: WO9200954A1] Compounds useful as inhibitors of retroviral proteases characterized by structure (I) wherein X<1> and X<2> may consist of 0-2 alpha -amino acid groups terminally substituted by hydrogen or one of a number of end groups, R<1>, R<2> can be selected from a wide variety of hydrocarbon radicals.

IPC 1-7

C07C 269/00; C07C 271/00; C07F 9/02

IPC 8 full level

A61K 38/55 (2006.01); A61P 31/12 (2006.01); C07F 9/30 (2006.01); C07F 9/32 (2006.01); C07F 9/38 (2006.01); C07F 9/40 (2006.01); C07K 1/113 (2006.01); C07K 5/06 (2006.01); C07K 14/81 (2006.01); A61K 38/00 (2006.01)

CPC (source: EP)

A61P 31/12 (2017.12); C07F 9/301 (2013.01); C07F 9/3211 (2013.01); C07K 5/06191 (2013.01); A61K 38/00 (2013.01)

Citation (search report)

  • [E] EP 0435059 A1 19910703 - HOECHST AG [DE]
  • [A] JOURNAL OF THE AMERICAN CHEMICAL SOCIETY vol. 106, no. 15, 25 July 1984, WASHINGTON, DC US pages 4282 - 4283 PAUL A. BARTLETT 'Phosphinic Acid Dipeptide Analogues: Potent, Slow-Binding Inhibitors of Aspartic Pepsidases'
  • See references of WO 9200954A1

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB GR IT LI LU NL SE

DOCDB simple family (publication)

WO 9200954 A1 19920123; AU 8191091 A 19920204; EP 0538374 A1 19930428; EP 0538374 A4 19930519; JP H05508846 A 19931209

DOCDB simple family (application)

US 9104759 W 19910703; AU 8191091 A 19910703; EP 91913442 A 19910703; JP 51231291 A 19910703