EP 0541757 A1 19930519 - NEW HETERO-ARYLOXY--g(b)-CARBOLINES, THEIR PREPARATION AND THEIR USE IN MEDICAMENTS.
Title (en)
NEW HETERO-ARYLOXY--g(b)-CARBOLINES, THEIR PREPARATION AND THEIR USE IN MEDICAMENTS.
Title (de)
NEUE HETARYLOXY--g(b)-CARBOLINE, DEREN HERSTELLUNG UND VERWENDUNG IN ARZNEIMITTELN.
Title (fr)
NOUVELLES HETARYLOXY--g(b)-CARBOLINES, LEUR FABRICATION ET LEUR UTILISATION DANS DES MEDICAMENTS.
Publication
Application
Priority
DE 4118741 A 19910605
Abstract (en)
[origin: WO9221679A1] Described are hetero-aryloxy-$g(b)-carbolines of the formula (I), in which R?A is a triazine-condensed or benzo-condensed heteroaryl entity with 1-2 nitrogen atoms, which may optionally be substituted by halogen, C1-6?alkyl, C1-6?alkoxy, C1-6?alkylthio, trifluoromethyl or SO2?-R?1, or a 5 or 6-membered hetero-aryl entity with 1-2 nitrogen atoms, substituted by halogen, C1-6?alkyl, C1-6?alkoxy, C1-6?alkylthio, trifluoromethyl or SO2?-R?1. Also described is the preparation of these compounds and their use in medicaments.
Abstract (fr)
Il est décrit des hétaryloxy-beta-carbolines ayant la formule (I) dans laquelle RA désigne un reste hétaryle condensé en triazine ou en benzène, avec 1 à 2 atomes d'azote, éventuellement substitué par un halogène, un alkyle en C1-6, un alcoxy en C1-6, un alkylthio en C1-6, un trifluorométhyle ou SO2-R1, ou encore un reste hétaryle à 5 ou 6 éléments, avec 1 à 2 atomes d'azote, substitué par un halogène, un alkyle en C1-6, un alcoxy en C1-6, un alkylthio en C1-6, un trifluorométhyle ou SO2-R1, ainsi que leur fabrication et leur utilisation dans des médicaments.
IPC 1-7
IPC 8 full level
A61K 31/435 (2006.01); A61K 31/44 (2006.01); A61K 31/47 (2006.01); A61K 31/50 (2006.01); A61K 31/505 (2006.01); A61P 25/02 (2006.01); A61P 25/08 (2006.01); A61P 25/20 (2006.01); C07D 471/04 (2006.01)
CPC (source: EP KR US)
A61P 25/02 (2017.12 - EP); A61P 25/08 (2017.12 - EP); A61P 25/20 (2017.12 - EP); C07D 471/04 (2013.01 - EP KR US)
Citation (search report)
See references of WO 9221679A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IT LI LU MC NL SE
DOCDB simple family (publication)
WO 9221679 A1 19921210; AU 1807492 A 19921210; AU 658631 B2 19950427; CA 2087098 A1 19921206; CN 1039906 C 19980923; CN 1069270 A 19930224; CZ 281810 B6 19970212; CZ 396892 A3 19931013; DE 4118741 A1 19921210; EP 0541757 A1 19930519; FI 930293 A0 19930125; FI 930293 A 19930125; HU 9300595 D0 19930528; HU T63166 A 19930728; IE 921825 A1 19921216; IL 102116 A0 19930114; IL 102116 A 19970218; JP H06500341 A 19940113; KR 930701440 A 19930611; MX 9202616 A 19930901; NO 300771 B1 19970721; NO 930390 D0 19930204; NO 930390 L 19930204; NZ 243014 A 19950427; PL 172481 B1 19970930; PL 297839 A1 19931102; PT 100565 A 19930831; RU 2105766 C1 19980227; US 5348958 A 19940920; US 5698555 A 19971216; ZA 924127 B 19930224
DOCDB simple family (application)
DE 9200465 W 19920604; AU 1807492 A 19920605; CA 2087098 A 19920604; CN 92105684 A 19920604; CS 396892 A 19920604; DE 4118741 A 19910605; EP 92911058 A 19920604; FI 930293 A 19930125; HU 9300595 A 19920604; IE 921825 A 19920701; IL 10211692 A 19920605; JP 50977492 A 19920604; KR 930700323 A 19930204; MX 9202616 A 19920602; NO 930390 A 19930204; NZ 24301492 A 19920604; PL 29783992 A 19920604; PT 10056592 A 19920604; RU 93005125 A 19930204; US 27246494 A 19940711; US 89281992 A 19920605; ZA 924127 A 19920605