EP 0552247 A1 19930728 - PEPTIDES CONTAINING SUBSTITUTED 1,4-DIAMINES AS TRANSITION-STATE INSERTS.
Title (en)
PEPTIDES CONTAINING SUBSTITUTED 1,4-DIAMINES AS TRANSITION-STATE INSERTS.
Title (de)
PEPTIDE MIT SUBSTITUIERTEN 1,4-DIAMINEN ALS ÜBERGANGSZUSTANDEINSCHUB.
Title (fr)
PEPTIDES CONTENANT DES 1,4-DIAMINES SUBSTITUEES COMME SEGMENTS D'INSERTION A L'ETAT DE TRANSITION.
Publication
Application
Priority
US 59547090 A 19901010
Abstract (en)
[origin: WO9206996A1] The present invention provides novel peptides of formula (I). These peptides are useful as inhibitors of retroviral proteases. Inhibitors of retroviral proteases, such as the HIV-I protease, are useful for treating diseases caused by retroviruses, such as human acquired immunodeficiency disease syndrome (AIDS).
Abstract (fr)
L'invention se rapporte à de nouveaux peptides représentés par la formule (I) et qui sont utiles comme inhibiteurs des protéases rétrovirales. Les inhibiteurs des protéases rétrovirales, comme la protéase du VIH-I, servent à traiter les maladies causées par les rétrovirus, telles que le syndrome immunodéficitaire acquis (SIDA) chez l'homme.
IPC 1-7
IPC 8 full level
A61K 31/13 (2006.01); A61K 31/215 (2006.01); A61K 31/40 (2006.01); A61K 31/42 (2006.01); A61K 31/425 (2006.01); A61K 38/00 (2006.01); A61P 31/12 (2006.01); A61P 31/18 (2006.01); C07C 237/22 (2006.01); C07C 271/20 (2006.01); C07C 271/22 (2006.01); C07D 233/26 (2006.01); C07K 5/02 (2006.01); C07K 5/06 (2006.01); C07K 14/81 (2006.01)
CPC (source: EP)
A61P 31/12 (2017.12); A61P 31/18 (2017.12); C07C 271/20 (2013.01); C07C 271/22 (2013.01); C07D 233/26 (2013.01); C07K 5/021 (2013.01); A61K 38/00 (2013.01)
Citation (search report)
See references of WO 9206996A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IT LI LU NL SE
DOCDB simple family (publication)
WO 9206996 A1 19920430; AU 8759491 A 19920520; EP 0552247 A1 19930728; JP H06502403 A 19940317
DOCDB simple family (application)
US 9107047 W 19911001; AU 8759491 A 19911001; EP 91918640 A 19911001; JP 51792391 A 19911001