EP 0575500 A4 19940601 - HIV PROTEASE INHIBITORS
Title (en)
HIV PROTEASE INHIBITORS
Publication
Application
Priority
US 66629291 A 19910308
Abstract (en)
[origin: WO9215319A1] The invention relates to HIV protease inhibitors wherein the compounds have a 2,4-dihydroxy isostere wherein the hydroxyl group in the 2-position is further substituted to create a tertiary alcohol. Also disclosed are pharmaceutically acceptable salts thereof, which inhibit HIV-I protease and are useful in the treatment of AIDS.
IPC 1-7
IPC 8 full level
A61K 31/16 (2006.01); A61K 31/19 (2006.01); A61K 31/195 (2006.01); A61K 31/22 (2006.01); A61P 31/12 (2006.01); A61P 31/18 (2006.01); A61P 37/04 (2006.01); A61P 43/00 (2006.01); C07C 221/00 (2006.01); C07C 225/02 (2006.01); C07C 233/30 (2006.01); C07C 233/47 (2006.01); C07C 237/12 (2006.01); C07C 237/22 (2006.01); C07C 271/06 (2006.01); C07C 271/22 (2006.01); C07C 311/32 (2006.01); C07K 5/02 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP)
A61P 31/12 (2017.12); A61P 31/18 (2017.12); A61P 37/04 (2017.12); A61P 43/00 (2017.12); C07C 237/22 (2013.01); C07C 271/22 (2013.01); C07K 5/0207 (2013.01); A61K 38/00 (2013.01)
Citation (search report)
- No further relevant documents disclosed
- See references of WO 9215319A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IT LI LU MC NL SE
DOCDB simple family (publication)
WO 9215319 A1 19920917; EP 0575500 A1 19931229; EP 0575500 A4 19940601; JP H06505495 A 19940623
DOCDB simple family (application)
US 9201738 W 19920307; EP 92908310 A 19920307; JP 50826393 A 19920307