EP 0581777 A1 19940209 - STEREOSELECTIVE PREPARATION OF SUBSTITUTED PIPERIDINES.
Title (en)
STEREOSELECTIVE PREPARATION OF SUBSTITUTED PIPERIDINES.
Title (de)
STEREOSELEKTIVE HERSTELLUNG VON SUBSTITUIERTEN PIPERIDINEN.
Title (fr)
PREPARATION STEREOSELECTIVE DE PIPERIDINES SUBSTITUEES.
Publication
Application
Priority
US 67524491 A 19910326
Abstract (en)
[origin: US5686615A] Novel processes are disclosed for the stereoselective preparation of substituted piperidine derivatives of the formulae <IMAGE> (IV) and <IMAGE> (I) wherein R1 and R2 are defined as below, useful as substance P receptor antagonists and in treating diseases mediated by an excess of substance P.
Abstract (fr)
Nouveaux procédés de préparation stéréosélective de dérivés de pipéridine substituée répondant aux formules (IV) et (I), dans lesquelles R1 et R2 ont les mêmes notations que ci-dessous.
IPC 1-7
IPC 8 full level
A61K 31/4427 (2006.01); A61K 31/443 (2006.01); A61K 31/4433 (2006.01); A61K 31/445 (2006.01); A61K 31/451 (2006.01); A61K 31/452 (2006.01); A61K 31/4523 (2006.01); A61K 31/47 (2006.01); A61P 3/00 (2006.01); A61P 9/08 (2006.01); A61P 9/10 (2006.01); A61P 17/00 (2006.01); A61P 25/00 (2006.01); A61P 25/02 (2006.01); A61P 29/00 (2006.01); A61P 37/08 (2006.01); C07B 53/00 (2006.01); C07C 45/44 (2006.01); C07C 45/51 (2006.01); C07C 45/67 (2006.01); C07C 45/71 (2006.01); C07C 47/565 (2006.01); C07C 47/575 (2006.01); C07C 205/44 (2006.01); C07D 211/56 (2006.01); C07D 401/12 (2006.01); C07D 405/12 (2006.01); C07D 409/04 (2006.01); C07D 409/12 (2006.01); C07D 409/14 (2006.01)
IPC 8 main group level
C07D (2006.01)
CPC (source: EP US)
A61P 3/00 (2017.12 - EP); A61P 9/08 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 17/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/02 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 37/08 (2017.12 - EP); C07C 45/44 (2013.01 - EP US); C07C 45/513 (2013.01 - EP US); C07C 45/673 (2013.01 - EP US); C07C 45/71 (2013.01 - EP US); C07C 47/565 (2013.01 - EP US); C07C 47/575 (2013.01 - EP US); C07D 211/56 (2013.01 - EP US); C07D 401/12 (2013.01 - EP US); C07D 409/12 (2013.01 - EP US); Y02P 20/55 (2015.11 - EP)
Citation (search report)
See references of WO 9217449A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IT LI LU NL SE
DOCDB simple family (publication)
US 5686615 A 19971111; AU 1244892 A 19921102; AU 647592 B2 19940324; BR 9205807 A 19940628; CA 2106200 A1 19920927; CA 2106200 C 19961119; CN 1038932 C 19980701; CN 1065264 A 19921014; CZ 289960 B6 20020515; CZ 293954 B6 20040818; CZ 293955 B6 20040818; CZ 367292 A3 19930915; EG 19976 A 19970130; EP 0581777 A1 19940209; FI 106199 B 20001215; FI 934186 A0 19930924; FI 934186 A 19930924; HU 9302709 D0 19931228; HU T67276 A 19950328; IE 920939 A1 19921007; IL 101328 A0 19921115; IL 101328 A 20001031; IL 137021 A0 20010614; JP H06502182 A 19940310; JP H0794440 B2 19951011; KR 0145432 B1 19980715; MX 9201315 A 19921001; MY 110886 A 19990630; NO 180484 B 19970120; NO 180484 C 19970430; NO 933413 D0 19930924; NO 933413 L 19930924; NZ 242116 A 19951026; PL 169993 B1 19960930; PT 100282 A 19930630; RU 2105001 C1 19980220; SK 284185 B6 20041005; SK 284565 B6 20050602; SK 367292 A3 20001211; TW 213900 B 19931001; WO 9217449 A1 19921015; YU 29892 A 19941228; YU 48260 B 19970930; ZA 922164 B 19930927
DOCDB simple family (application)
US 11914993 A 19930920; AU 1244892 A 19920114; BR 9205807 A 19920114; CA 2106200 A 19920114; CN 92102009 A 19920325; CS 367292 A 19920114; CZ 387697 A 19920114; CZ 387797 A 19920114; EG 16092 A 19920326; EP 92905084 A 19920114; FI 934186 A 19930924; HU 9302709 A 19920114; IE 920939 A 19920325; IL 10132892 A 19920322; IL 13702100 A 20000626; JP 50474792 A 19920114; KR 930702889 A 19930925; MX 9201315 A 19920324; MY PI19920521 A 19920326; NO 933413 A 19930924; NZ 24211692 A 19920325; PL 30111092 A 19920114; PT 10028292 A 19920324; RU 93057733 A 19920114; SK 367292 A 19920114; SK 99699 A 19920114; TW 81100889 A 19920210; US 9200065 W 19920114; YU 29892 A 19920325; ZA 922164 A 19920325