EP 0638080 A4 19950823 - 7-DISUBSTITUTED-METHYL-4-OXO-3H -,5H --PYRROLO 3,2-d -]PYRIMIDINE AND PHARMACEUTICAL USES AND COMPOSITIONS CONTAINING THE SAME.
Title (en)
7-DISUBSTITUTED-METHYL-4-OXO-3H -,5H --PYRROLO 3,2-d -]PYRIMIDINE AND PHARMACEUTICAL USES AND COMPOSITIONS CONTAINING THE SAME.
Title (de)
7-DISUBSTITUIERTE-METHYL-4-OXO-3H, 5H-PYRROLO-(3,2-d) PYRIMIDINDERIVATE, DEREN PHARMAZEUTISCHE VERWENDUNG UND DIESE VERBINDUNGEN ENTHALTENDE ZUSAMMENSETZUNGEN.
Title (fr)
PYRIMIDINE 7-BISUBSTITUEE-METHYL-4-OXO-3H -, 5H --PYRROLO 3,2-d -], UTILISATION PHARMACEUTIQUE ET COMPOSITIONS CONTENANT LADITE PYRIMIDINE.
Publication
Application
Priority
- US 9302841 W 19930325
- US 87144192 A 19920421
Abstract (en)
[origin: WO9321187A1] Disclosed is a compound of formula (I) where R<1> is H, NH2, or OCH3, R<2> is an optionally substituted cyclic group optionally containing one or more heteroatoms, R<3> and R<4> are independently H or C1-4 alkyl, m is 0-4, n is 0-6, p is 0.1, X is CN, CSNH2, PO(OH)2, COOH, SO2NH2, NH2, OH, CNHNH2, tetrazole, triazole, or COR<5> where R<5> is C1-4 alkyl, CF3, NH2, or OC1-4 alkyl, and Y is O or NH that is useful as a pharmaceutical.
IPC 1-7
C07D 487/04; C07D 265/30; C07D 237/08; C07D 241/12; C07D 213/57; C07D 233/64; C07D 277/30; C07D 207/337; C07D 207/34; C07D 333/24; C07D 307/81
IPC 8 full level
A61K 31/505 (2006.01); A61P 31/12 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07C 255/31 (2006.01); C07C 255/35 (2006.01); C07C 255/40 (2006.01); C07C 255/42 (2006.01); C07D 207/34 (2006.01); C07D 487/04 (2006.01); C07F 9/6561 (2006.01)
CPC (source: EP KR)
A61P 31/12 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07C 255/35 (2013.01 - EP); C07C 255/40 (2013.01 - EP); C07C 255/42 (2013.01 - EP KR); C07D 207/34 (2013.01 - EP KR); C07D 487/04 (2013.01 - EP KR); C07F 9/6561 (2013.01 - EP)
Citation (search report)
- No further relevant documents disclosed
- See references of WO 9321187A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9321187 A1 19931028; AU 4276693 A 19931118; CA 2133346 A1 19931028; EP 0638080 A1 19950215; EP 0638080 A4 19950823; FI 944933 A0 19941020; FI 944933 A 19941020; HU 9403021 D0 19941228; HU T71559 A 19951228; JP H07507062 A 19950803; KR 950701335 A 19950323; NO 303637 B1 19980810; NO 943988 D0 19941020; NO 943988 L 19941020; RU 94046387 A 19960927
DOCDB simple family (application)
US 9302841 W 19930325; AU 4276693 A 19930325; CA 2133346 A 19930325; EP 93912081 A 19930325; FI 944933 A 19941020; HU 9403021 A 19930325; JP 51835793 A 19930325; KR 19940703788 A 19941020; NO 943988 A 19941020; RU 94046387 A 19941118