Global Patent Index - EP 0641311 A1

EP 0641311 A1 19950308 - NOVEL DIHYDROXYBENZYLAMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME.

Title (en)

NOVEL DIHYDROXYBENZYLAMINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME.

Title (de)

DIHYDROXYBENZYL DERIVATE, DEREN HERSTELLUNG UND DEREN PHARMAZEUTISCHE ZUSAMMENSETZUNGEN.

Title (fr)

NOUVEAUX DERIVES DE LA DIHYDROXYBENZYLAMINE, LEUR PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES QUI LES CONTIENNENT.

Publication

EP 0641311 A1 19950308 (FR)

Application

EP 93910121 A 19930514

Priority

  • FR 9300468 W 19930514
  • FR 9205980 A 19920518

Abstract (en)

[origin: FR2691145A1] Novel 2,5 dihydroxybenzylamine derivatives of general formula (I), their preparation and pharmaceutical compositions containing same. In general formula (I), one of the symbols R1 or R2 denots a hydrogen or halo atom or a hydroxy, alkoxy, alkylcarbonyloxy arylcarbonyloxy, mercapto, alkylthio, amino, formylamino, alkylcarbonylamino, arylcarbonylamino radical and the other denotes an alkoxy, alkoxymethyl, acyl, arylcarbonyl, alkyloxycarbonyl, aryloxycarbonyl, alkenyloxycarbonyl, carbamoyl or thiocarbamoyl radical, the nitrogen atom being optionally substituted by one or two alkyl or phenyl radicals, the alkyl, phenyl and aryl radicals being optionally substituted. The novel products of formula (I) have outstanding tumour prevention activity.

IPC 1-7

C07C 229/64; C07C 229/60; C07C 237/30; C07C 237/44; A61K 31/135; A61K 31/165; C07C 225/22; C07C 327/48

IPC 8 full level

C07B 61/00 (2006.01); C07C 215/76 (2006.01); C07C 215/78 (2006.01); C07C 219/34 (2006.01); C07C 225/22 (2006.01); C07C 229/60 (2006.01); C07C 229/64 (2006.01); C07C 237/30 (2006.01); C07C 237/44 (2006.01); C07C 323/34 (2006.01); C07C 323/35 (2006.01); C07C 327/48 (2006.01)

CPC (source: EP)

C07C 229/64 (2013.01); C07C 237/44 (2013.01)

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

FR 2691145 A1 19931119; AU 4075693 A 19931213; EP 0641311 A1 19950308; JP H07506585 A 19950720; MX 9302869 A 19931101; TW 252095 B 19950721; WO 9323364 A1 19931125; ZA 933426 B 19940802

DOCDB simple family (application)

FR 9205980 A 19920518; AU 4075693 A 19930514; EP 93910121 A 19930514; FR 9300468 W 19930514; JP 51994493 A 19930514; MX 9302869 A 19930517; TW 82103887 A 19930518; ZA 933426 A 19930517