Global Patent Index - EP 0676959 A4

EP 0676959 A4 19960103 - ENDOTHELIN RECEPTOR ANTAGONISTS.

Title (en)

ENDOTHELIN RECEPTOR ANTAGONISTS.

Title (de)

ENDOTHELINREZEPTORANTAGONISTEN.

Title (fr)

ANTAGONISTES DES RECEPTEURS DE L'ENDOTHELINE.

Publication

EP 0676959 A4 19960103 (EN)

Application

EP 94904877 A 19931221

Priority

  • US 9312435 W 19931221
  • US 99546692 A 19921222

Abstract (en)

[origin: WO9414434A1] Indole derivatives of formula (1) wherein the substituents are defined herein are disclosed. The compounds are useful in methods of antagonizing endothelin receptors, treating hypertension, treating renal failure and treating cerebrovascular disease. Pharmaceutical compositions are also disclosed.

IPC 1-7

A61K 31/40; A61K 31/405; C07D 209/12; C07D 209/22; C07D 405/10; C07D 405/14

IPC 8 full level

A61K 31/40 (2006.01); A61K 31/403 (2006.01); A61K 31/404 (2006.01); A61P 9/00 (2006.01); A61P 9/12 (2006.01); A61P 13/02 (2006.01); A61P 15/00 (2006.01); A61P 43/00 (2006.01); C07D 209/30 (2006.01); C07D 405/04 (2006.01); C07D 405/06 (2006.01)

CPC (source: EP)

A61P 9/00 (2017.12); A61P 9/12 (2017.12); A61P 13/02 (2017.12); A61P 15/00 (2017.12); A61P 43/00 (2017.12); C07D 405/04 (2013.01); C07D 405/06 (2013.01)

Citation (search report)

Designated contracting state (EPC)

BE CH DE FR GB IT LI NL

DOCDB simple family (publication)

WO 9414434 A1 19940707; AU 5873594 A 19940719; CN 1096513 A 19941221; EP 0676959 A1 19951018; EP 0676959 A4 19960103; JP H08504826 A 19960528; MX 9400071 A 19940729; ZA 939516 B 19940606

DOCDB simple family (application)

US 9312435 W 19931221; AU 5873594 A 19931221; CN 93119929 A 19931222; EP 94904877 A 19931221; JP 51538694 A 19931221; MX 9400071 A 19940103; ZA 939516 A 19931220