EP 0679084 A1 19951102 - HYDANTOIN AND SUCCINIMIDE-SUBSTITUTED DERIVATIVES OF SPIROINDANYLCAMPHORSULFONYL OXYTOCIN ANTAGONISTS.
Title (en)
HYDANTOIN AND SUCCINIMIDE-SUBSTITUTED DERIVATIVES OF SPIROINDANYLCAMPHORSULFONYL OXYTOCIN ANTAGONISTS.
Title (de)
HYDRANTOIN- UND BERNSTEINSÄUREIMIDE-SUBSTITUIERTE DERIVATE VON SPIROINDANYLCAMPFERSULFINYL-OXYTOCIN-ANTAGONISTEN.
Title (fr)
DERIVES SUBSTITUES PAR SUCCINIMIDE ET HYDANTOINE, D'ANTAGONISTES D'OXYTOCINE DE SPIROINDANYLCAMPHROSULFONYLE.
Publication
Application
Priority
- US 9312565 W 19931223
- US 99386192 A 19921223
Abstract (en)
[origin: WO9414438A1] Compounds of formula (I) where X is (a) or (b), R is Het, wherein Het is as defined in the description. These compounds are oxytocin and vasopressin antagonists useful in the treatment of preterm labor, dysmenorrhea, and for the stoppage of labor preparatory to cesarean delivery, timing of parturition, uterine hyperactivity, endometriosis, hypertension, congestive heart failure, hyponatremia and cognitive disorders.
IPC 1-7
A61K 31/435; A61K 31/495; C07D 401/12; C07D 471/00; C07D 207/40; C07D 401/14
IPC 8 full level
C07D 295/22 (2006.01); A61K 31/4427 (2006.01); A61K 31/443 (2006.01); A61K 31/445 (2006.01); A61K 31/495 (2006.01); A61P 13/02 (2006.01); A61P 15/00 (2006.01); C07D 207/27 (2006.01); C07D 207/273 (2006.01); C07D 207/40 (2006.01); C07D 207/416 (2006.01); C07D 221/20 (2006.01); C07D 295/26 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 403/14 (2006.01); C07D 405/06 (2006.01); C07D 405/14 (2006.01); C07D 471/10 (2006.01); C07D 487/04 (2006.01); C07D 498/04 (2006.01); C07F 9/6558 (2006.01)
CPC (source: EP)
A61P 13/02 (2017.12); A61P 15/00 (2017.12); C07D 207/416 (2013.01); C07D 295/26 (2013.01); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 405/06 (2013.01); C07D 471/10 (2013.01); C07D 487/04 (2013.01); C07F 9/65583 (2013.01)
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9414438 A1 19940707; AU 5960194 A 19940719; AU 690534 B2 19980430; CA 2151821 A1 19940707; EP 0679084 A1 19951102; EP 0679084 A4 19951108; JP H08505150 A 19960604
DOCDB simple family (application)
US 9312565 W 19931223; AU 5960194 A 19931223; CA 2151821 A 19931223; EP 94905516 A 19931223; JP 51545994 A 19931223