Title (en)

NOVEL N-ARYLALIPHATIC-N-ALKYL-FUNCTIONALISED AMIDES, METHOD FOR THEIR PREPATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

Title (de)

N-ARYLALIPHATISCHE-N-ALKYLFUNKTIONALISIERTE AMIDE, VERFAHREN ZU IHRER HERSTELLUNG UND DIESE ENTHALTENDE PHARMAZEUTISCHE ZUBEREITUNGEN

Title (fr)

NOUVEAUX AMIDES N-ARYLALIPHATIQUES-N-ALKYL-FONCTIONNALISES, PROCEDE POUR LEUR PREPARATION ET COMPOSITIONS PHARMACEUTIQUES EN CONTENANT

Publication

EP 0700382 A1 19960313 (FR)

Application

EP 95914415 A 19950324

Priority

• FR 9500369 W 19950324
• FR 9403560 A 19940325

Abstract (en)

[origin: WO9526335A1] Novel n-arylaliphatic-n-alkyl-functionalised amides of formula (I), wherein Am is in particular a substituted piperidyl group. A method for preparing these compounds, and pharmaceutical compositions containing them are also disclosed. The compounds are neurokinin receptor antagonists.

IPC 1-7

C07D 211/14; A61K 31/445

IPC 8 full level

C07D 295/18 (2006.01); A61K 31/396 (2006.01); A61K 31/397 (2006.01); A61K 31/445 (2006.01); A61K 31/4468 (2006.01); A61K 31/451 (2006.01); A61P 43/00 (2006.01); C07D 211/14 (2006.01); C07D 211/52 (2006.01); C07D 211/58 (2006.01); C07D 239/26 (2006.01); C07D 453/02 (2006.01); C07D 455/02 (2006.01); C07D 471/04 (2006.01); C07D 477/00 (2006.01); C07D 487/04 (2006.01); C07D 487/08 (2006.01)

CPC (source: EP)

A61P 43/00 (2017.12); C07D 211/14 (2013.01); C07D 211/52 (2013.01); C07D 211/58 (2013.01)

Citation (search report)

See references of WO 9526335A1

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9526335 A1 19951005; AU 2142295 A 19951017; EP 0700382 A1 19960313; FR 2717802 A1 19950929; FR 2717802 B1 19960621; HU 9503366 D0 19960228; HU T73226 A 19960729; JP H08511277 A 19961126

DOCDB simple family (application)

FR 9500369 W 19950324; AU 2142295 A 19950324; EP 95914415 A 19950324; FR 9403560 A 19940325; HU 9503366 A 19950324; JP 52500395 A 19950324