EP 0711286 A1 19960515 - BENZOXAZINONES AND BENZOTHIAZINONES ENDOWED WITH THERAPEUTIC ACTIVITY

Title (en)

BENZOXAZINONES AND BENZOTHIAZINONES ENDOWED WITH THERAPEUTIC ACTIVITY

Title (de)

BENZOXAZINONE UND BENZOTHIAZINONE MIT THERAPEUTISCHER WIRKUNG

Title (fr)

BENZOXAZINONES ET BENZOTHIAZINONES AYANT UNE ACTIVITE THERAPEUTIQUE

Publication

EP 0711286 A1 19960515 (EN)

Application

EP 94924778 A 19940718

Priority

EP 9402354 W 19940718
IT MI931678 A 19930728

Abstract (en)

[origin: WO9504048A1] Compounds of general formula (I) wherein X is an oxygen or sulfur atom; Y is alkylene or cycloalkylene; A is hydroxy, alkoxy, acyloxy, mercapto, alkyl-sulfonyloxy, phenyl-sulfonyloxy, (a) or (b) wherein R3 is an alkyl or alkylene group omega -substituted by 2,3-dihydro-4H-1,3-benzoxazin-4-one-N-yl; R is hydrogen, alkyl or phenyl; R1 and R2 are independently hydrogen, halogen, alkoxy, trifluoromethyl or alkyl; and the pharmaceutically acceptable acid and base salts thereof, are useful as therapeutically active substances.

IPC 1-7

C07D 265/22; C07D 279/08; A61K 31/535; A61K 31/54

IPC 8 full level

A61K 31/535 (2006.01); A61K 31/536 (2006.01); A61K 31/54 (2006.01); A61K 31/5415 (2006.01); A61P 9/08 (2006.01); A61P 9/10 (2006.01); C07D 265/22 (2006.01); C07D 279/08 (2006.01); C07D 417/06 (2006.01); C07D 417/08 (2006.01)

CPC (source: EP)

A61P 9/08 (2018.01); A61P 9/10 (2018.01); C07D 265/22 (2013.01); C07D 279/08 (2013.01)

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9504048 A1 19950209; AU 7494594 A 19950228; CA 2168099 A1 19950209; CN 1128025 A 19960731; EP 0711286 A1 19960515; FI 960342 A0 19960125; FI 960342 A 19960125; HU 9600165 D0 19960328; HU T74587 A 19970128; IL 110473 A0 19941021; IT 1264812 B1 19961010; IT MI931678 A0 19930728; IT MI931678 A1 19950128; JP H09500878 A 19970128; NO 960308 D0 19960125; NO 960308 L 19960313; TW 277061 B 19960601; ZA 945555 B 19950303

DOCDB simple family (application)

EP 9402354 W 19940718; AU 7494594 A 19940718; CA 2168099 A 19940718; CN 94192889 A 19940718; EP 94924778 A 19940718; FI 960342 A 19960125; HU 9600165 A 19940718; IL 11047394 A 19940727; IT MI931678 A 19930728; JP 50552995 A 19940718; NO 960308 A 19960125; TW 83106854 A 19940727; ZA 945555 A 19940727