EP 0717622 A4 19980909 - METHODS OF TREATING HIV WITH AZASPIRANES
Title (en)
METHODS OF TREATING HIV WITH AZASPIRANES
Title (de)
VERFAHREN ZUR BEHANDLUNG VON HIV MIT AZASPIRANEN
Title (fr)
PROCEDES DE TRAITEMENT DU VIH AU MOYEN D'AZASPIRANES
Publication
Application
Priority
- GB 9315351 A 19930723
- US 9408274 W 19940722
Abstract (en)
[origin: WO9503049A1] Invented is a method for inhibiting cellular entry of human immunodeficiency viruses (HIV) in HIV seropositive humans which comprises administering to such human an effective amount of a substituted azaspirane.
IPC 1-7
IPC 8 full level
C07D 221/20 (2006.01); A61K 31/40 (2006.01); A61K 31/403 (2006.01); A61K 31/435 (2006.01); A61P 31/12 (2006.01); A61P 37/04 (2006.01); C07D 209/54 (2006.01)
CPC (source: EP)
A61K 31/40 (2013.01); A61K 31/435 (2013.01); A61P 31/12 (2017.12); A61P 37/04 (2017.12)
Citation (search report)
- [E] WO 9503041 A1 19950202 - SMITHKLINE BEECHAM CORP [US], et al
- [E] WO 9503042 A1 19950202 - SMITHKLINE BEECHAM CORP [US], et al
- [E] WO 9503047 A1 19950202 - SMITHKLINE BEECHAM CORP [US], et al
- [PX] WO 9314760 A2 19930805 - SMITHKLINE BEECHAM CORP [US]
- [PX] WO 9315735 A1 19930819 - SMITHKLINE BEECHAM CORP [US]
- [X] WO 9214462 A1 19920903 - SMITHKLINE BEECHAM CORP [US]
- [Y] BADGER A M ET AL: "ANTIARTHRITIC AND SUPPRESSOR CELL INDUCING ACTIVITY OF AZASPIRANES:STRUCTURE-FUNCTION RELATIONSHIPS OF A NOVEL CLASS OF IMMUNOMODULATORY AGENTS", JOURNAL OF MEDICINAL CHEMISTRY, vol. 33, no. 11, November 1990 (1990-11-01), pages 2963 - 2970, XP000605424
- [Y] S. GOODMAN: "THERAPEUTIC EFFECTS OF ORGANIC GERMANIUM", MEDICAL HYPOTHESES, vol. 26, 1988, pages 207 - 215, XP002069578
- [Y] P.S. SARIN ET AL.: "INHIBITION OF HTLV-III REPLICTION IN CELL CULTURES", NATO ASI SER., SER. A, vol. 120, 1986, pages 329 - 342, XP002069579
- See references of WO 9503049A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9503049 A1 19950202; AU 7514094 A 19950220; CA 2167843 A1 19950202; CN 1130873 A 19960911; EP 0717622 A1 19960626; EP 0717622 A4 19980909; GB 9315351 D0 19930908; JP H09500646 A 19970121; NZ 271496 A 19990629; ZA 945417 B 19950510
DOCDB simple family (application)
US 9408274 W 19940722; AU 7514094 A 19940722; CA 2167843 A 19940722; CN 94193382 A 19940722; EP 94925100 A 19940722; GB 9315351 A 19930723; JP 50533095 A 19940722; NZ 27149694 A 19940722; ZA 945417 A 19940722