Global Patent Index - EP 0717622 A4

EP 0717622 A4 19980909 - METHODS OF TREATING HIV WITH AZASPIRANES

Title (en)

METHODS OF TREATING HIV WITH AZASPIRANES

Title (de)

VERFAHREN ZUR BEHANDLUNG VON HIV MIT AZASPIRANEN

Title (fr)

PROCEDES DE TRAITEMENT DU VIH AU MOYEN D'AZASPIRANES

Publication

EP 0717622 A4 19980909 (EN)

Application

EP 94925100 A 19940722

Priority

  • GB 9315351 A 19930723
  • US 9408274 W 19940722

Abstract (en)

[origin: WO9503049A1] Invented is a method for inhibiting cellular entry of human immunodeficiency viruses (HIV) in HIV seropositive humans which comprises administering to such human an effective amount of a substituted azaspirane.

IPC 1-7

A61K 31/44; A61K 31/40

IPC 8 full level

C07D 221/20 (2006.01); A61K 31/40 (2006.01); A61K 31/403 (2006.01); A61K 31/435 (2006.01); A61P 31/12 (2006.01); A61P 37/04 (2006.01); C07D 209/54 (2006.01)

CPC (source: EP)

A61K 31/40 (2013.01); A61K 31/435 (2013.01); A61P 31/12 (2017.12); A61P 37/04 (2017.12)

Citation (search report)

  • [E] WO 9503041 A1 19950202 - SMITHKLINE BEECHAM CORP [US], et al
  • [E] WO 9503042 A1 19950202 - SMITHKLINE BEECHAM CORP [US], et al
  • [E] WO 9503047 A1 19950202 - SMITHKLINE BEECHAM CORP [US], et al
  • [PX] WO 9314760 A2 19930805 - SMITHKLINE BEECHAM CORP [US]
  • [PX] WO 9315735 A1 19930819 - SMITHKLINE BEECHAM CORP [US]
  • [X] WO 9214462 A1 19920903 - SMITHKLINE BEECHAM CORP [US]
  • [Y] BADGER A M ET AL: "ANTIARTHRITIC AND SUPPRESSOR CELL INDUCING ACTIVITY OF AZASPIRANES:STRUCTURE-FUNCTION RELATIONSHIPS OF A NOVEL CLASS OF IMMUNOMODULATORY AGENTS", JOURNAL OF MEDICINAL CHEMISTRY, vol. 33, no. 11, November 1990 (1990-11-01), pages 2963 - 2970, XP000605424
  • [Y] S. GOODMAN: "THERAPEUTIC EFFECTS OF ORGANIC GERMANIUM", MEDICAL HYPOTHESES, vol. 26, 1988, pages 207 - 215, XP002069578
  • [Y] P.S. SARIN ET AL.: "INHIBITION OF HTLV-III REPLICTION IN CELL CULTURES", NATO ASI SER., SER. A, vol. 120, 1986, pages 329 - 342, XP002069579
  • See references of WO 9503049A1

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9503049 A1 19950202; AU 7514094 A 19950220; CA 2167843 A1 19950202; CN 1130873 A 19960911; EP 0717622 A1 19960626; EP 0717622 A4 19980909; GB 9315351 D0 19930908; JP H09500646 A 19970121; NZ 271496 A 19990629; ZA 945417 B 19950510

DOCDB simple family (application)

US 9408274 W 19940722; AU 7514094 A 19940722; CA 2167843 A 19940722; CN 94193382 A 19940722; EP 94925100 A 19940722; GB 9315351 A 19930723; JP 50533095 A 19940722; NZ 27149694 A 19940722; ZA 945417 A 19940722