EP 0730605 A1 19960911 - SUBSTITUTED DI- AND TRIPEPTIDE INHIBITORS OF PROTEIN:FARNESYL TRANSFERASE
Title (en)
SUBSTITUTED DI- AND TRIPEPTIDE INHIBITORS OF PROTEIN:FARNESYL TRANSFERASE
Title (de)
SUBSTITUIERTE DI- UND TRIPEPTIDE MIT PROTEIN: FARNESYL TRANSFERASE INHIBIERENDE AKTIVITÄT
Title (fr)
INHIBITEURS DI- ET TRIPEPTIDIQUES SUBSTITUES DE L'ENZYME PROTEINE:LA FARNESYLE TRANSFERASE
Publication
Application
Priority
- US 9411553 W 19941012
- US 14873593 A 19931105
- US 30330194 A 19940913
Abstract (en)
[origin: WO9512612A1] Novel inhibitors of protein:farnesyl transferase enzyme are described, as well as methods for the preparation and pharmaceutical compositions of the same, which are useful in controlling tissue proliferative diseases, including cancer and restenosis.
IPC 1-7
IPC 8 full level
A61K 38/55 (2006.01); A61P 9/00 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07K 5/078 (2006.01); C07K 5/097 (2006.01); C12N 9/99 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP)
A61P 9/00 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07K 5/06147 (2013.01); A61K 38/00 (2013.01)
Citation (search report)
See references of WO 9512612A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9512612 A1 19950511; AU 681454 B2 19970828; AU 7976094 A 19950523; CA 2170766 A1 19950511; EP 0730605 A1 19960911; FI 961819 A0 19960429; FI 961819 A 19960429; HU 9601193 D0 19960729; HU T75308 A 19970528; JP 3597863 B2 20041208; JP H09504547 A 19970506; KR 100362338 B1 20030408; NO 961814 D0 19960503; NO 961814 L 19960506; NZ 275691 A 19980325
DOCDB simple family (application)
US 9411553 W 19941012; AU 7976094 A 19941012; CA 2170766 A 19941012; EP 94930725 A 19941012; FI 961819 A 19960429; HU 9601193 A 19941012; JP 51322495 A 19941012; KR 19960702309 A 19960503; NO 961814 A 19960503; NZ 27569194 A 19941012