EP 0748333 A4 20000510 - ANTITHROMBOTIC AGENTS
Title (en)
ANTITHROMBOTIC AGENTS
Title (de)
ANTITHROMBOTISCHE STOFFE
Title (fr)
AGENTS ANTITHROMBOTIQUES
Publication
Application
Priority
- US 20650094 A 19940304
- US 31860094 A 19941005
- US 9502627 W 19950303
Abstract (en)
[origin: WO9523809A1] This invention relates to L-arginine aldehyde derivatives having formula (I) where R<1>, X and Y have the values defined in the description, as well as pharmaceutical formulations containing those compounds and methods of their use as thrombin inhibitors, coagulation inhibitors and thromboembolic disorder agents.
IPC 1-7
C07K 5/00; C07K 7/00; C07K 17/00; A61K 38/00; C07D 417/00; C07D 279/10; C07D 279/12; C07D 295/00; C07D 413/00; C07D 237/00; C07D 237/02
IPC 8 full level
A61K 31/40 (2006.01); A61K 31/42 (2006.01); A61K 31/425 (2006.01); A61K 31/44 (2006.01); A61K 31/4427 (2006.01); A61K 31/47 (2006.01); A61K 38/55 (2006.01); A61P 7/02 (2006.01); C07D 207/16 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01); C07D 413/12 (2006.01); C07D 417/12 (2006.01); C07K 5/065 (2006.01); C07K 5/078 (2006.01); C07K 5/083 (2006.01); C07K 5/087 (2006.01); C07K 14/47 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP)
A61P 7/02 (2017.12); C07K 5/06078 (2013.01); C07K 5/06139 (2013.01); A61K 38/00 (2013.01)
Citation (search report)
- [X] EP 0526877 A2 19930210 - BRISTOL MYERS SQUIBB CO [US]
- [X] US 5250660 A 19931005 - SHUMAN ROBERT T [US]
- [A] EP 0479489 A2 19920408 - LILLY CO ELI [US]
- [A] EP 0542525 A2 19930519 - LILLY CO ELI [US]
- [E] EP 0643073 A1 19950315 - LILLY CO ELI [US]
- See references of WO 9523809A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9523809 A1 19950908; AU 1884395 A 19950918; CA 2184188 A1 19950908; EP 0748333 A1 19961218; EP 0748333 A4 20000510; JP H09509943 A 19971007
DOCDB simple family (application)
US 9502627 W 19950303; AU 1884395 A 19950303; CA 2184188 A 19950303; EP 95911134 A 19950303; JP 52304095 A 19950303