Global patent index - EP 0748333 A4

EP 0748333 A4 2000-05-10 - ANTITHROMBOTIC AGENTS

Title (en)

ANTITHROMBOTIC AGENTS

Title (de)

ANTITHROMBOTISCHE STOFFE

Title (fr)

AGENTS ANTITHROMBOTIQUES

Publication

EP 0748333 A4 (EN)

Application

EP 95911134 A

Priority

  • US 20650094 A
  • US 31860094 A
  • US 9502627 W

Abstract (en)

[origin: WO9523809A1] This invention relates to L-arginine aldehyde derivatives having formula (I) where R<1>, X and Y have the values defined in the description, as well as pharmaceutical formulations containing those compounds and methods of their use as thrombin inhibitors, coagulation inhibitors and thromboembolic disorder agents.

IPC 1-7 (main, further and additional classification)

C07K 5/00; A61K 38/00; C07D 237/00; C07D 237/02; C07D 279/10; C07D 279/12; C07D 295/00; C07D 413/00; C07D 417/00; C07K 7/00; C07K 17/00

IPC 8 full level (invention and additional information)

C07D 401/12 (2006.01); A61K 31/40 (2006.01); A61K 31/42 (2006.01); A61K 31/425 (2006.01); A61K 31/44 (2006.01); A61K 31/4427 (2006.01); A61K 31/47 (2006.01); A61K 38/55 (2006.01); A61P 7/02 (2006.01); C07D 207/16 (2006.01); C07D 403/12 (2006.01); C07D 413/12 (2006.01); C07D 417/12 (2006.01); C07K 5/065 (2006.01); C07K 5/078 (2006.01); C07K 5/083 (2006.01); C07K 5/087 (2006.01); C07K 14/47 (2006.01); A61K 38/00 (2006.01)

CPC (invention and additional information)

C07K 5/06139 (2013.01); C07K 5/06078 (2013.01); A61K 38/00 (2013.01)

Citation (search report)

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9523809 A1 19950908; AU 1884395 A 19950918; CA 2184188 A1 19950908; EP 0748333 A1 19961218; EP 0748333 A4 20000510; JP H09509943 A 19971007

INPADOC legal status

2004-04-07 [18D] DEEMED TO BE WITHDRAWN

- Ref Legal Event Code: 18D

- Effective date: 20031001

2004-01-21 [17Q] FIRST EXAMINATION REPORT

- Ref Legal Event Code: 17Q

- Effective date: 20031209

2000-05-10 [A4] SUPPLEMENTARY SEARCH REPORT

- Ref Legal Event Code: A4

- Effective date: 20000328

2000-05-10 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

1996-12-18 [17P] REQUEST FOR EXAMINATION FILED

- Ref Legal Event Code: 17P

- Effective date: 19960830

1996-12-18 [AK] DESIGNATED CONTRACTING STATES:

- Ref Legal Event Code: AK

- Designated State(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

1996-12-18 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Ref Legal Event Code: AX

- Free Format Text: LT PAYMENT 960830;SI PAYMENT 960830