EP 0785937 A1 19970730 - 2-(IMIDAZOL-4-YL)CARBAPENEME DERIVATIVES, INTERMEDIATES THEREOF AND USE AS ANTIBACTERIALS
Title (en)
2-(IMIDAZOL-4-YL)CARBAPENEME DERIVATIVES, INTERMEDIATES THEREOF AND USE AS ANTIBACTERIALS
Title (de)
2-(IMIDAZOL-4-YL)CARBAPENEMDERIVATE, IHRE ZWISCHENPRODUKTE UND VERWENDUNG ALS ANTIBAKTERIELLE MITTEL
Title (fr)
DERIVES DE 2-(IMIDAZOL-4-YL)CARBAPENEME, LEURS INTERMEDIAIRES AINSI QUE LEUR UTILISATION EN TANT QU'ANTIBACTERIENS
Publication
Application
Priority
- EP 9503888 W 19951002
- GB 9420710 A 19941014
- GB 9424248 A 19941201
Abstract (en)
[origin: WO9611932A1] Compounds of general formula (I), in which R<a> or R<b> alone is hydrogen, optionally substituted (C1-6)alkyl or together form a 5 or 6 membered heterocyclic ring which may contain at least one additional heteroatom selected from oxygen, nitrogen or sulphur; R<1> is (C1-6)alkyl which is unsubstituted or substituted by fluoro, a hydroxy group which is optionally protected by a readily removable hydroxy protecting group, or by an amino group which is optionally protected by a readily removable amino protecting group; R<2> is hydrogen or methyl and -CO2R<3> is carboxy or a carboxylate anion or the group R<3> is a readily removable carboxy protecting group, are useful in the treatment and prophylaxis of bacterial infections in animals and humans.
IPC 1-7
IPC 8 full level
A61K 31/397 (2006.01); A61K 31/415 (2006.01); A61P 31/04 (2006.01); C07D 403/06 (2006.01); C07D 477/00 (2006.01); C07D 477/14 (2006.01)
CPC (source: EP)
A61P 31/04 (2017.12); C07D 403/06 (2013.01); C07D 477/14 (2013.01); Y02P 20/55 (2015.11)
Citation (search report)
See references of WO 9611932A1
Designated contracting state (EPC)
AT BE CH DE DK FR GB IT LI NL SE
DOCDB simple family (publication)
WO 9611932 A1 19960425; EP 0785937 A1 19970730; JP H10507185 A 19980714
DOCDB simple family (application)
EP 9503888 W 19951002; EP 95934654 A 19951002; JP 51288896 A 19951002