EP 0786997 A4 19980311 - MUSCARINE ANTAGONISTS
Title (en)
MUSCARINE ANTAGONISTS
Title (de)
MUSCARINANTAGONISTEN
Title (fr)
ANTAGONISTES DE MUSCARINE
Publication
Application
Priority
- US 9513710 W 19951024
- US 32975794 A 19941027
- US 44015395 A 19950512
Abstract (en)
[origin: WO9613262A1] Compounds, 1,3-dihydro-1-{1-[piperidin-4-yl]piperidin-4-yl}-2H-benzimidazol-2-ones and 1,3-dihydro-1-{4-amino-1-cyclohexyl}-2H-benzimidazol-2-ones and derivatives thereof, their preparation, method of use and pharmaceutical compositions are described. These compounds are endowed with antimuscarinic activity and are useful in the treatment and/or prevention of myopia (commonly known as nearsightedness).
IPC 1-7
A61K 31/415; A61K 31/42; A61K 31/425; A61K 31/445; A61K 31/44; A61K 31/505; A61K 31/495; A61K 31/33; C07D 243/04; C07D 233/04; C07D 263/62
IPC 8 full level
A61K 31/454 (2006.01); A61K 31/4545 (2006.01); A61K 31/497 (2006.01); A61K 31/501 (2006.01); A61K 31/506 (2006.01); A61K 31/522 (2006.01); A61K 31/5377 (2006.01); A61P 27/02 (2006.01); A61P 43/00 (2006.01); C07D 401/04 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 403/12 (2006.01); C07D 471/04 (2006.01)
CPC (source: EP)
A61P 27/02 (2017.12); A61P 43/00 (2017.12); C07D 401/04 (2013.01); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 403/12 (2013.01)
Citation (search report)
- [X] US 4329353 A 19820511 - STOKBROEKX RAYMOND A, et al
- See references of WO 9613262A1
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9613262 A1 19960509; AU 3967495 A 19960523; AU 701127 B2 19990121; CA 2200468 A1 19960509; EP 0786997 A1 19970806; EP 0786997 A4 19980311; JP 2002515008 A 20020521
DOCDB simple family (application)
US 9513710 W 19951024; AU 3967495 A 19951024; CA 2200468 A 19951024; EP 95937615 A 19951024; JP 51469196 A 19951024