EP 0799188 B1 19990915 - AMIDES OF MONO AND DICARBOXYLIC ACIDS WITH GLYCOSAMINES, SELECTIVELY ACTIVE ON THE CANNABINOID PERIPHERAL RECEPTOR
Title (en)
AMIDES OF MONO AND DICARBOXYLIC ACIDS WITH GLYCOSAMINES, SELECTIVELY ACTIVE ON THE CANNABINOID PERIPHERAL RECEPTOR
Title (de)
AMIDE VON MONO-UND DICARBONSÄUREN MIT GLYCOSAMINEN, MIT SELEKTIVER WIRKUNG AUF DEN PERIPHEREN CANNABINOIDEN REZEPTOR
Title (fr)
AMIDES D'ACIDES MONO ET BICARBOXYLIQUES A GLYCOSAMINES, A ACTIVITE SELECTIVE SUR LE RECEPTEUR PERIPHERIQUE DES CANNABINOIDES
Publication
Application
Priority
- EP 9504926 W 19951213
- IT MI942513 A 19941214
Abstract (en)
[origin: WO9618600A1] The vast number of theoretically conceivable compounds resulting from the combination of all claimed substituents in formula (I) precludes a comprehensive search. For economical reasons the search has been limited to the following compounds: R1 is a hydrocarbon radical unsubstituted or substituted by only one OH-group and having a linear chain of at least 8 carbons atoms(A); the NR2R3 group is either a linear alpha-, beta-, or gamma-, amino acid (e.g. amino acids like proline are not included), or a glycosamine residue. Despite the above limitation the search revealed too many relevant compounds. Therefore the search was further limited to compounds with NR2R3 = Glycine, beta-Alamine, gamma-amino-butyric acid, Serine- or Cysteine derivatives, or glycosamine of the following structures: (a), (b), (c). Still too many pertinent compounds where retrieved which can not all be cited in the search report. The documents cited are only an arbitrary selection and the search report has to be regarded as incomplete.
IPC 1-7
C07C 233/47; C07C 323/59; C07H 13/06; C07D 207/16; A61K 31/195; A61K 31/22; A61K 31/70; A61K 31/40
IPC 8 full level
A61K 31/70 (2006.01); A61K 31/7024 (2006.01); A61P 9/08 (2006.01); A61P 9/10 (2006.01); A61P 11/00 (2006.01); A61P 25/00 (2006.01); A61P 25/08 (2006.01); A61P 25/28 (2006.01); A61P 27/00 (2006.01); A61P 27/02 (2006.01); A61P 29/00 (2006.01); A61P 31/12 (2006.01); A61P 37/00 (2006.01); A61P 37/04 (2006.01); C07C 233/18 (2006.01); C07C 233/20 (2006.01); C07C 233/47 (2006.01); C07C 233/49 (2006.01); C07C 323/59 (2006.01); C07D 207/16 (2006.01); C07H 13/06 (2006.01)
CPC (source: EP)
A61P 9/08 (2018.01); A61P 9/10 (2018.01); A61P 11/00 (2018.01); A61P 25/00 (2018.01); A61P 25/08 (2018.01); A61P 25/28 (2018.01); A61P 27/00 (2018.01); A61P 27/02 (2018.01); A61P 29/00 (2018.01); A61P 31/12 (2018.01); A61P 37/00 (2018.01); A61P 37/04 (2018.01); C07C 233/18 (2013.01); C07C 233/20 (2013.01); C07C 233/47 (2013.01); C07C 233/49 (2013.01); C07C 323/59 (2013.01); C07D 207/16 (2013.01); C07H 13/06 (2013.01)
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9618600 A1 19960620; AT E184591 T1 19991015; AU 4344196 A 19960703; CA 2207804 A1 19960620; CA 2207804 C 20070807; DE 69512273 D1 19991021; DE 69512273 T2 20000511; EP 0799188 A2 19971008; EP 0799188 B1 19990915; IL 116401 A0 19960331; IT 1271267 B 19970527; IT MI942513 A0 19941214; IT MI942513 A1 19960614; JP 4111349 B2 20080702; JP H11501615 A 19990209
DOCDB simple family (application)
EP 9504926 W 19951213; AT 95942141 T 19951213; AU 4344196 A 19951213; CA 2207804 A 19951213; DE 69512273 T 19951213; EP 95942141 A 19951213; IL 11640195 A 19951214; IT MI942513 A 19941214; JP 51826496 A 19951213