EP 0804420 A1 19971105 - TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS
Title (en)
TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS
Title (de)
TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS
Title (fr)
BENZAZEPINE TRICYCLE ANTAGONISTE DE LA VASOPRESSINE
Publication
Application
Priority
- US 9601051 W 19960116
- US 37316995 A 19950117
- US 54880595 A 19951222
Abstract (en)
[origin: WO9622282A1] Tricyclic compound of general formula (I) as defined herein which exhibit antagonist activity at V1 and/or V2 receptors and exhibit in vivo vasopressin antagonist activity, methods for using such compounds in treating diseases characterized by excess renal reabsorption of water, and process for preparing such compounds.
IPC 1-7
C07D 223/20; C07D 223/28; C07D 401/12; C07D 495/04; A61K 31/55; C07D 487/04; C07D 498/04; C07D 267/20; C07D 243/38; C07D 471/04
IPC 8 full level
A61K 31/55 (2006.01); A61P 13/02 (2006.01); A61P 15/00 (2006.01); A61P 43/00 (2006.01); C07D 223/20 (2006.01); C07D 223/28 (2006.01); C07D 243/38 (2006.01); C07D 267/16 (2006.01); C07D 267/20 (2006.01); C07D 401/06 (2006.01); C07D 401/12 (2006.01); C07D 405/06 (2006.01); C07D 405/12 (2006.01); C07D 405/14 (2006.01); C07D 409/12 (2006.01); C07D 413/06 (2006.01); C07D 413/14 (2006.01); C07D 471/04 (2006.01); C07D 487/04 (2006.01); C07D 495/04 (2006.01); C07D 498/04 (2006.01); C07D 513/04 (2006.01)
CPC (source: EP)
A61P 9/00 (2018.01); A61P 13/02 (2018.01); A61P 15/00 (2018.01); A61P 15/06 (2018.01); A61P 43/00 (2018.01); C07D 223/20 (2013.01); C07D 223/28 (2013.01); C07D 243/38 (2013.01); C07D 267/20 (2013.01); C07D 401/12 (2013.01); C07D 471/04 (2013.01); C07D 487/04 (2013.01); C07D 495/04 (2013.01)
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9622282 A1 19960725; AR 002459 A1 19980325; AU 4904296 A 19960807; BR 9606977 A 19971104; CA 2210688 A1 19960725; CN 1190391 A 19980812; CZ 224597 A3 19971217; EA 000752 B1 20000424; EA 199700116 A1 19971230; EP 0804420 A1 19971105; HU P9801219 A2 19981028; HU P9801219 A3 20000728; IL 116777 A0 19960514; IL 116777 A 20001121; JP H10512865 A 19981208; NZ 302881 A 19990329; TW 449584 B 20010811
DOCDB simple family (application)
US 9601051 W 19960116; AR 10102796 A 19960115; AU 4904296 A 19960116; BR 9606977 A 19960116; CA 2210688 A 19960116; CN 96192568 A 19960116; CZ 224597 A 19960116; EA 199700116 A 19960116; EP 96905227 A 19960116; HU P9801219 A 19960116; IL 11677796 A 19960116; JP 52244896 A 19960116; NZ 30288196 A 19960116; TW 85100462 A 19960116