EP 0804463 A1 19971105 - NEUROKININE (TACHYKININE) ANTAGONISTS
Title (en)
NEUROKININE (TACHYKININE) ANTAGONISTS
Title (de)
NEUROKININ (TACHYKININ)-ANTAGONISTEN
Title (fr)
ANTAGONISTES DE LA NEUROKININE (TACHYKININE)
Publication
Application
Priority
- DE 4416255 A 19940507
- DE 4445939 A 19941222
- EP 9501691 W 19950504
Abstract (en)
[origin: US5700827A] The invention relates to new amino acid derivatives of general formula I R1-R11-A1B(I) and the pharmaceutically acceptable salts thereof, wherein group B is -A2-NR2R3 or R5, and wherein R1, A1, A2, R2, R3, R5 and R11 have the meanings described in the specification, as well as the preparation and use thereof. The novel compounds are valuable neurokinin (tachykinin) antagonists.
IPC 1-7
IPC 8 full level
A61K 38/00 (2006.01); A61K 38/05 (2006.01); A61P 1/04 (2006.01); A61P 11/00 (2006.01); A61P 25/18 (2006.01); A61P 25/28 (2006.01); A61P 27/02 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07K 5/06 (2006.01); C07K 5/078 (2006.01); C07K 5/097 (2006.01)
CPC (source: EP US)
A61P 1/04 (2018.01 - EP); A61P 11/00 (2018.01 - EP); A61P 25/18 (2018.01 - EP); A61P 25/28 (2018.01 - EP); A61P 27/02 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 35/00 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07K 5/06139 (2013.01 - EP US); C07K 5/06165 (2013.01 - EP US); C07K 5/0821 (2013.01 - EP US); A61K 38/00 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
US 5700827 A 19971223; AU 2524995 A 19951129; AU 690275 B2 19980423; BG 100946 A 19970731; CA 2189764 A1 19951116; CN 1147260 A 19970409; CZ 325496 A3 19970917; EE 9600186 A 19970815; EP 0804463 A1 19971105; FI 964473 A0 19961107; FI 964473 A 19961107; HR P950276 A2 19970430; HU 9603082 D0 19970128; HU T75708 A 19970528; IL 113625 A0 19950831; JP H09512806 A 19971222; MX 9605128 A 19970830; NO 964700 D0 19961106; NO 964700 L 19961106; NZ 285750 A 19980826; PL 317127 A1 19970317; RO 115355 B1 20000128; SK 142696 A3 19970604; US 5712273 A 19980127; WO 9530687 A1 19951116
DOCDB simple family (application)
US 47527895 A 19950607; AU 2524995 A 19950504; BG 10094696 A 19961029; CA 2189764 A 19950504; CN 95192859 A 19950504; CZ 325496 A 19950504; EE 9600186 A 19950504; EP 9501691 W 19950504; EP 95919392 A 19950504; FI 964473 A 19961107; HR P950276 A 19950505; HU 9603082 A 19950504; IL 11362595 A 19950505; JP 52867795 A 19950504; MX 9605128 A 19950504; NO 964700 A 19961106; NZ 28575095 A 19950504; PL 31712795 A 19950504; RO 9602085 A 19950504; SK 142696 A 19950504; US 43461395 A 19950504