Global Patent Index - EP 0845987 A4

EP 0845987 A4 20000524 - C-PROTEINASE INHIBITORS FOR THE TREATMENT OF DISORDERS RELATED TO THE OVERPRODUCTION OF COLLAGEN

Title (en)

C-PROTEINASE INHIBITORS FOR THE TREATMENT OF DISORDERS RELATED TO THE OVERPRODUCTION OF COLLAGEN

Title (de)

C - PROTEINASEINHIBITOREN ZUR BEHANDLUNG VON STÖRUNGEN, DIE MIT EINER KOLLAGENÜBERPRODUKTION ZUSAMMENHÄNGEN

Title (fr)

INHIBITEURS DE LA C-PROTEINASE DESTINES AU TRAITEMENT DES AFFECTIONS LIEES A LA SURPRODUCTION DE COLLAGENE

Publication

EP 0845987 A4 20000524 (EN)

Application

EP 96930499 A 19960808

Priority

  • US 9612876 W 19960808
  • US 203895 P 19950808
  • US 60120396 A 19960214
  • US 60918796 A 19960301

Abstract (en)

[origin: WO9705865A1] The present invention relates to the novel use of organic molecules capable of inhibiting C-proteinase activity in order to regulate, modulate and/or inhibit abnormal collagen formation.

IPC 1-7

A61K 31/215; A61K 31/38; A61K 31/40; A61K 31/66; A61K 31/165; A61K 31/70; A61K 31/34; C07C 259/06; C07C 311/29; C07D 207/48; C07C 323/60; C07K 5/02; C07F 9/40

IPC 8 full level

A61K 31/00 (2006.01); A61K 31/40 (2006.01); A61K 38/00 (2006.01); A61P 1/00 (2006.01); A61P 1/16 (2006.01); A61P 5/24 (2006.01); A61P 11/00 (2006.01); A61P 13/00 (2006.01); A61P 13/12 (2006.01); A61P 17/00 (2006.01); A61P 43/00 (2006.01); C07C 259/06 (2006.01); C07C 311/19 (2006.01); C07C 311/29 (2006.01); C07C 323/60 (2006.01); C07D 207/48 (2006.01); C07F 9/24 (2006.01); C07F 9/40 (2006.01); C07K 5/02 (2006.01); C07K 5/072 (2006.01)

CPC (source: EP KR)

A61K 31/215 (2013.01 - KR); A61P 1/00 (2017.12 - EP); A61P 1/16 (2017.12 - EP); A61P 5/24 (2017.12 - EP); A61P 11/00 (2017.12 - EP); A61P 13/00 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 17/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07C 259/06 (2013.01 - EP); C07C 311/29 (2013.01 - EP); C07C 323/60 (2013.01 - EP); C07D 207/48 (2013.01 - EP); C07F 9/4006 (2013.01 - EP); C07K 5/022 (2013.01 - EP)

Citation (search report)

  • [X] EP 0606046 A1 19940713 - CIBA GEIGY AG [CH]
  • [X] US 4687841 A 19870818 - SPILBURG CURTIS A [US], et al
  • [X] WO 9115507 A1 19911017 - BEECHAM GROUP PLC [GB]
  • [X] EP 0262399 A2 19880406 - TAKEDA CHEMICAL INDUSTRIES LTD [JP]
  • [X] CHEMICAL ABSTRACTS, vol. 113, no. 17, 22 October 1990, Columbus, Ohio, US; abstract no. 147795, ODAKE, SHINJIRO ET AL: "Vertebrate collagenase inhibitor. I. Tripeptidyl hydroxamic acids" XP002134085 & CHEM. PHARM. BULL. ( 1990 ), 38(4), 1007-11, 1990
  • [X] CHEMICAL ABSTRACTS, vol. 110, no. 23, 5 June 1989, Columbus, Ohio, US; abstract no. 205068, LELIEVRE, Y. ET AL: "Synovial collagenase inhibition by actinonin. Structure-activity relations" XP002134086 & PATHOL. BIOL. ( 1989 ), 37(1), 43-6, 1989
  • [X] BRINGMANN, GERHARD ET AL: "Acetogenic isoquinoline alkaloids. 66. First total synthesis of korupensamines A and B", HETEROCYCLES ( 1994 ), 39(2), 503-8, 1994, XP000561812
  • [X] CHEMICAL ABSTRACTS, vol. 123, no. 23, 4 December 1995, Columbus, Ohio, US; abstract no. 314466, OUCHI, T. ET AL: "Synthesis of polydepsipeptide with pendant carboxylic acid groups and its hydrolysis behavior" XP002134087 & STUD. POLYM. SCI. ( 1994 ), 12(BIODEGRADABLE PLASTICS AND POLYMERS), 528-33, 1994
  • [X] CHEMICAL ABSTRACTS, vol. 116, no. 17, 27 April 1992, Columbus, Ohio, US; abstract no. 174753, PERICH, JOHN W. ET AL: "Synthesis of casein-related peptides and phosphopeptides. XVI. The efficient synthesis of the casein-related O-phosphoseryl-containing peptide Ac-Glu-Ser(P)-Leu-Ser(P)-Ser(P)-Ser(P)-Glu-Glu-NHMe" XP002134088 & AUST. J. CHEM. ( 1992 ), 45(2), 385-94, 1992
  • See references of WO 9705865A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9705865 A1 19970220; AU 6951296 A 19970305; BR 9609883 A 19990323; CA 2229098 A1 19970220; CN 1198096 A 19981104; EP 0845987 A1 19980610; EP 0845987 A4 20000524; JP H11511137 A 19990928; KR 19990036271 A 19990525; MX 9801093 A 19980430

DOCDB simple family (application)

US 9612876 W 19960808; AU 6951296 A 19960808; BR 9609883 A 19960808; CA 2229098 A 19960808; CN 96197271 A 19960808; EP 96930499 A 19960808; JP 50864897 A 19960808; KR 19980700939 A 19980209; MX 9801093 A 19960808