Global Patent Index - EP 0856000 A1

EP 0856000 A1 19980805 - 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION

Title (en)

1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION

Title (de)

1,3,5-TRISUBSTITUIERTE PYRAZOLE ZUR BEHANDLUNG VON ENTZÜNDUNGEN

Title (fr)

PYRAZOLES 1,3,5-TRISUBSTITUES POUR LE TRAITEMENT DES INFLAMMATIONS

Publication

EP 0856000 A1 19980805 (EN)

Application

EP 96932841 A 19961008

Priority

  • GB 9520584 A 19951009
  • JP 9602919 W 19961008

Abstract (en)

[origin: WO9713755A1] A compound of the formula (I) wherein R<1> is hydroxyethyl, 1-hydroxy-1-methylethyl, hydrogen, halogen, nitro, or cyano, R<2> is chloro, cyano, or lower alkyl optionally substituted with halogen, and R<3> is lower alkylthio, lower alkylsulfinyl, or lower alkylsulfonyl, provided that when R<1> is hydrogen, halogen, nitro, or cyano, then R<2> is chloro, and a pharmaceutically acceptable salt thereof, processes for their preparation and pharmaceutical compositions.

IPC 1-7

C07D 231/12; C07D 231/14; A61K 31/415; C07D 231/16

IPC 8 full level

A61K 31/00 (2006.01); A61K 31/415 (2006.01); A61P 29/00 (2006.01); C07D 231/12 (2006.01); C07D 231/14 (2006.01); C07D 231/16 (2006.01)

CPC (source: EP KR)

A61K 31/415 (2013.01 - KR); A61P 29/00 (2017.12 - EP); C07D 231/12 (2013.01 - EP KR); C07D 231/14 (2013.01 - EP KR); C07D 231/16 (2013.01 - EP KR)

Citation (search report)

See references of WO 9713755A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9713755 A1 19970417; AU 7146196 A 19970430; CA 2234511 A1 19970417; CN 1203589 A 19981230; EP 0856000 A1 19980805; GB 9520584 D0 19951213; JP H11513403 A 19991116; KR 19990063989 A 19990726; ZA 968286 B 19970513

DOCDB simple family (application)

JP 9602919 W 19961008; AU 7146196 A 19961008; CA 2234511 A 19961008; CN 96198649 A 19961008; EP 96932841 A 19961008; GB 9520584 A 19951009; JP 51490997 A 19961008; KR 19980702464 A 19980403; ZA 968286 A 19961002