Global Patent Index - EP 0869943 A1

EP 0869943 A1 19981014 - MONOCYCLIC BETA-LACTAME DERIVATIVES FOR TREATMENT OF ATHEROSCLEROSIS

Title (en)

MONOCYCLIC BETA-LACTAME DERIVATIVES FOR TREATMENT OF ATHEROSCLEROSIS

Title (de)

MONOCYCLISCHE BETA-LACTAME ZUR BEHANDLUNG VON ATHEROSKLEROSE

Title (fr)

DERIVES DE BETA-LACTAME MONOCYCLIQUES UTILISES DANS LE TRAITEMENT DE L'ATHEROSCLEROSE

Publication

EP 0869943 A1 19981014 (EN)

Application

EP 96943110 A 19961204

Priority

  • EP 9605587 W 19961204
  • GB 9525131 A 19951208
  • GB 9623756 A 19961115

Abstract (en)

[origin: WO9721675A1] Compounds of formula (I) are prodrugs of the corresponding compounds in which CO2R<3> is CO2H. These are inhibitors of the phospholipase A2 enzyme Lp-PLA2 and of use in treating atherosclerosis.

IPC 1-7

C07D 205/09; A61K 31/395; C07D 205/08; C07D 405/12

IPC 8 full level

A61K 31/00 (2006.01); A61K 31/395 (2006.01); A61K 31/397 (2006.01); A61P 3/00 (2006.01); A61P 3/10 (2006.01); A61P 9/00 (2006.01); A61P 9/10 (2006.01); A61P 19/00 (2006.01); A61P 19/02 (2006.01); A61P 25/18 (2006.01); A61P 29/00 (2006.01); A61P 43/00 (2006.01); C07D 205/08 (2006.01); C07D 205/09 (2006.01); C07D 405/12 (2006.01)

CPC (source: EP)

A61P 3/00 (2017.12); A61P 3/10 (2017.12); A61P 9/00 (2017.12); A61P 9/10 (2017.12); A61P 19/00 (2017.12); A61P 19/02 (2017.12); A61P 25/18 (2017.12); A61P 29/00 (2017.12); A61P 43/00 (2017.12); C07D 205/08 (2013.01); C07D 205/09 (2013.01); C07D 405/12 (2013.01)

Citation (search report)

See references of WO 9721675A1

Designated contracting state (EPC)

BE CH DE ES FR GB IT LI NL

DOCDB simple family (publication)

WO 9721675 A1 19970619; EP 0869943 A1 19981014; JP 2000502079 A 20000222

DOCDB simple family (application)

EP 9605587 W 19961204; EP 96943110 A 19961204; JP 52174697 A 19961204