EP 0869943 A1 19981014 - MONOCYCLIC BETA-LACTAME DERIVATIVES FOR TREATMENT OF ATHEROSCLEROSIS
Title (en)
MONOCYCLIC BETA-LACTAME DERIVATIVES FOR TREATMENT OF ATHEROSCLEROSIS
Title (de)
MONOCYCLISCHE BETA-LACTAME ZUR BEHANDLUNG VON ATHEROSKLEROSE
Title (fr)
DERIVES DE BETA-LACTAME MONOCYCLIQUES UTILISES DANS LE TRAITEMENT DE L'ATHEROSCLEROSE
Publication
Application
Priority
- EP 9605587 W 19961204
- GB 9525131 A 19951208
- GB 9623756 A 19961115
Abstract (en)
[origin: WO9721675A1] Compounds of formula (I) are prodrugs of the corresponding compounds in which CO2R<3> is CO2H. These are inhibitors of the phospholipase A2 enzyme Lp-PLA2 and of use in treating atherosclerosis.
IPC 1-7
IPC 8 full level
A61K 31/00 (2006.01); A61K 31/395 (2006.01); A61K 31/397 (2006.01); A61P 3/00 (2006.01); A61P 3/10 (2006.01); A61P 9/00 (2006.01); A61P 9/10 (2006.01); A61P 19/00 (2006.01); A61P 19/02 (2006.01); A61P 25/18 (2006.01); A61P 29/00 (2006.01); A61P 43/00 (2006.01); C07D 205/08 (2006.01); C07D 205/09 (2006.01); C07D 405/12 (2006.01)
CPC (source: EP)
A61P 3/00 (2017.12); A61P 3/10 (2017.12); A61P 9/00 (2017.12); A61P 9/10 (2017.12); A61P 19/00 (2017.12); A61P 19/02 (2017.12); A61P 25/18 (2017.12); A61P 29/00 (2017.12); A61P 43/00 (2017.12); C07D 205/08 (2013.01); C07D 205/09 (2013.01); C07D 405/12 (2013.01)
Citation (search report)
See references of WO 9721675A1
Designated contracting state (EPC)
BE CH DE ES FR GB IT LI NL
DOCDB simple family (publication)
WO 9721675 A1 19970619; EP 0869943 A1 19981014; JP 2000502079 A 20000222
DOCDB simple family (application)
EP 9605587 W 19961204; EP 96943110 A 19961204; JP 52174697 A 19961204