EP 0871628 A1 19981021 - QUINOLIZINONE TYPE COMPOUNDS
Title (en)
QUINOLIZINONE TYPE COMPOUNDS
Title (de)
VERBINDUNGEN DES CHINOLIZINON-TYPS
Title (fr)
COMPOSES DE TYPE QUINOLIZINONE
Publication
Application
Priority
- US 46915995 A 19950606
- US 63811296 A 19960529
- US 9608991 W 19960605
Abstract (en)
[origin: WO9639407A1] Antibacterial compounds having formula (I) and the pharmaceutically acceptable salts, esters and amides thereof, selected preferred examples of which include those compounds wherein A is =CR<6>-; R<1> is cycloalkyl of from three to eight carbon atoms or substituted phenyl; R<2> is selected from the group consisting of (a), (b), (c) and (d); R<3> is halogen; R<4> is hydrogen, loweralkyl, a pharmaceutically acceptable cation, or a prodrug ester group; R<5> is hydrogen, loweralkyl, halo(loweralkyl), or -NR<13>R<14>; and R<6> is halogen, loeralkyl, halo(loweralkyl), hydroxy-substituted loweralkyl, loweralkoxy(loweralkyl), loweralkoxy, or amino(loweralkyl), as well as pharmaceutical compositions containing such compounds and the use of the same in the treatment of bacterial infections.
IPC 1-7
C07D 471/04; C07D 455/02; C07D 491/16; C07D 519/00; A61K 31/435; A61K 31/505; C07D 213/68; C07D 213/61
IPC 8 full level
A61K 31/00 (2006.01); A61K 31/44 (2006.01); A61K 31/505 (2006.01); A61K 31/519 (2006.01); A61K 31/529 (2006.01); A61P 31/00 (2006.01); A61P 31/04 (2006.01); C07D 213/61 (2006.01); C07D 213/68 (2006.01); C07D 455/02 (2006.01); C07D 471/04 (2006.01); C07D 491/16 (2006.01); C07D 495/16 (2006.01); C07D 519/00 (2006.01); C07K 5/06 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP)
A61P 31/00 (2017.12); A61P 31/04 (2017.12); C07D 213/61 (2013.01); C07D 213/68 (2013.01); C07D 455/02 (2013.01); C07D 471/04 (2013.01); C07K 5/06026 (2013.01); A61K 38/00 (2013.01)
Citation (search report)
See references of WO 9639407A1
Designated contracting state (EPC)
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9639407 A1 19961212; AU 6153096 A 19961224; CA 2222322 A1 19961212; EP 0871628 A1 19981021; IL 122296 A0 19980405; JP H11510478 A 19990914; KR 19990022524 A 19990325; MX 9709416 A 19980731
DOCDB simple family (application)
US 9608991 W 19960605; AU 6153096 A 19960605; CA 2222322 A 19960605; EP 96919103 A 19960605; IL 12229696 A 19960605; JP 50142097 A 19960605; KR 19970709005 A 19971206; MX 9709416 A 19971202