Global Patent Index - EP 0885226 A1

EP 0885226 A1 19981223 - 4-AMINO PYRIMIDINE DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION

Title (en)

4-AMINO PYRIMIDINE DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION

Title (de)

4-AMINO-PYRIMIDIN-DERIVATE, DIESE VERBINDUNGEN ENTHALTENDE ARZNEIMITTEL, DEREN VERWENDUNG UND VERFAHREN ZU IHRER HERSTELLUNG

Title (fr)

DERIVES DE 4-AMINO-PYRIMIDINE, MEDICAMENTS CONTENANT CES COMPOSES, LEUR UTILISATION ET LEUR PROCEDE DE PRODUCTION

Publication

EP 0885226 A1 19981223 (DE)

Application

EP 97907066 A 19970303

Priority

  • DE 19608631 A 19960306
  • DE 19629652 A 19960723
  • EP 9701057 W 19970303

Abstract (en)

[origin: WO9732881A1] The present invention relates to 4-amino pyrimidine derivatives of general formula (I), where Ra, Rb, A and B are as defined in claim 1, their tautomers, stereoisomers and salts, especially their physiologically acceptable salts with inorganic or organic acids or bases, having valuable pharmacological properties, especially an inhibitory effect on signal transduction produced by tyrosinkinases, their use in the treatment of disorders, especially tumours, and their production.

IPC 1-7

C07D 487/04; C07D 471/04; A61K 31/505

IPC 8 full level

A61K 31/00 (2006.01); A61K 31/505 (2006.01); A61K 31/519 (2006.01); A61K 31/529 (2006.01); A61K 31/535 (2006.01); A61K 31/5375 (2006.01); A61K 31/5377 (2006.01); A61P 17/00 (2006.01); A61P 17/06 (2006.01); A61P 35/00 (2006.01); A61P 37/00 (2006.01); A61P 43/00 (2006.01); C07D 471/04 (2006.01); C07D 487/04 (2006.01); C07D 519/00 (2006.01)

CPC (source: EP KR)

A61P 17/00 (2018.01 - EP); A61P 17/06 (2018.01 - EP); A61P 35/00 (2018.01 - EP); A61P 37/00 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07D 471/04 (2013.01 - EP KR); C07D 487/04 (2013.01 - EP)

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9732881 A1 19970912; AU 1925197 A 19970922; AU 710274 B2 19990916; BG 102708 A 19990930; BR 9708312 A 19990803; CA 2243994 A1 19970912; CN 1212695 A 19990331; CZ 281798 A3 19990217; DE 19629652 A1 19980129; EE 9800277 A 19990215; EP 0885226 A1 19981223; HU P9901820 A2 19990928; HU P9901820 A3 20011029; IL 125404 A0 19990312; JP 2000506847 A 20000606; KR 19990087550 A 19991227; NO 984084 D0 19980904; NO 984084 L 19980904; NZ 331546 A 20000327; PL 328771 A1 19990215; SK 120598 A3 19990611; TR 199801749 T2 19981221

DOCDB simple family (application)

EP 9701057 W 19970303; AU 1925197 A 19970303; BG 10270898 A 19980820; BR 9708312 A 19970303; CA 2243994 A 19970303; CN 97192787 A 19970303; CZ 281798 A 19970303; DE 19629652 A 19960723; EE 9800277 A 19970303; EP 97907066 A 19970303; HU P9901820 A 19970303; IL 12540497 A 19970303; JP 53144497 A 19970303; KR 19980706987 A 19980905; NO 984084 A 19980904; NZ 33154697 A 19970303; PL 32877197 A 19970303; SK 120598 A 19970303; TR 9801749 T 19970303