Global Patent Index - EP 0894003 A1

EP 0894003 A1 19990203 - N-FORMYL HYDROXYLAMINE CONTAINING COMPOUNDS USEFUL AS ACE INHIBITORS AND/OR NEP INHIBITORS

Title (en)

N-FORMYL HYDROXYLAMINE CONTAINING COMPOUNDS USEFUL AS ACE INHIBITORS AND/OR NEP INHIBITORS

Title (de)

N-Formyl Hydroxylamin enthaltende Verbindungen als ACE und/oder NEP Inhibitoren

Title (fr)

COMPOSES A BASE DE N-FORMYL HYDROXYLAMINE CONVENANT COMME INHIBITEURS DE L'ENZYME ACE ET/OU DE L'ENDOPEPTIDASE NEP

Publication

EP 0894003 A1 19990203 (EN)

Application

EP 97917889 A 19970407

Priority

  • US 9705744 W 19970407
  • US 1629596 P 19960412

Abstract (en)

[origin: WO9738705A1] N-formyl hydroxylamines are provided which have structure (I) wherein R and R<1> are as defined herein and A is a dipeptide derived from an amino acid or is a conformationally restricted dipeptide mimic.

IPC 1-7

A61K 38/05

IPC 8 full level

C07D 233/10 (2006.01); A61K 31/00 (2006.01); A61K 31/195 (2006.01); A61K 31/198 (2006.01); A61K 31/435 (2006.01); A61K 31/4353 (2006.01); A61K 31/4365 (2006.01); A61K 31/55 (2006.01); A61K 31/551 (2006.01); A61K 31/553 (2006.01); A61K 38/00 (2006.01); A61P 9/00 (2006.01); A61P 9/12 (2006.01); A61P 43/00 (2006.01); C07C 259/06 (2006.01); C07D 267/14 (2006.01); C07D 471/04 (2006.01); C07D 471/06 (2006.01); C07D 487/04 (2006.01); C07D 495/14 (2006.01); C07D 498/04 (2006.01); C07D 513/04 (2006.01); C07K 5/02 (2006.01); C07K 5/023 (2006.01)

CPC (source: EP)

A61P 9/00 (2017.12); A61P 9/12 (2017.12); A61P 43/00 (2017.12); C07K 5/0202 (2013.01); A61K 38/00 (2013.01)

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9738705 A1 19971023; AU 2609497 A 19971107; AU 715451 B2 20000203; CA 2251292 A1 19971023; EP 0894003 A1 19990203; EP 0894003 A4 20001004; JP 2000511882 A 20000912

DOCDB simple family (application)

US 9705744 W 19970407; AU 2609497 A 19970407; CA 2251292 A 19970407; EP 97917889 A 19970407; JP 53716897 A 19970407