Global Patent Index - EP 0898564 A1

EP 0898564 A1 19990303 - METHOD OF PREPARING PHOSPHODIESTERASE IV INHIBITORS

Title (en)

METHOD OF PREPARING PHOSPHODIESTERASE IV INHIBITORS

Title (de)

VERFAHREN ZUR HERSTELLUNG VON PHOSPHORODIESTERASE-IV-HEMMERN

Title (fr)

PROCEDE DE PREPARATION D'INHIBITEURS DE PHOSPHODIESTERASE IV

Publication

EP 0898564 A1 19990303 (EN)

Application

EP 97920379 A 19970414

Priority

  • GB 9612083 A 19960610
  • US 9706131 W 19970414
  • US 1568796 P 19960417

Abstract (en)

[origin: WO9738976A1] A process for the preparation of a compound of structural formula (1) wherein R<1> is alkyl, alkenyl, phenyl or substituted phenyl, which comprises the addition of R<1> to an intermediate 2: by treatment of 2 with (R<1>)3M followed by reductive removal of the sulfinyl group.

IPC 1-7

C07D 213/30; C07D 213/34; A61K 31/44

IPC 8 full level

C07D 213/34 (2006.01)

CPC (source: EP)

A61P 11/06 (2017.12); C07D 213/34 (2013.01)

Citation (search report)

See references of WO 9738976A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9738976 A1 19971023; AR 006550 A1 19990908; AU 2459297 A 19971107; BR 9708684 A 19990803; CN 1216532 A 19990512; CZ 333298 A3 19990317; EA 000877 B1 20000626; EA 199800931 A1 19990429; EP 0898564 A1 19990303; SK 143198 A3 19990611; TW 426669 B 20010321

DOCDB simple family (application)

US 9706131 W 19970414; AR P970101372 A 19970407; AU 2459297 A 19970414; BR 9708684 A 19970414; CN 97193932 A 19970414; CZ 333298 A 19970414; EA 199800931 A 19970414; EP 97920379 A 19970414; SK 143198 A 19970414; TW 86104869 A 19970415