Global Patent Index - EP 0912090 A4

EP 0912090 A4 20000517 - INSECTICIDAL N-(SUBSTITUTED ARYLMETHYL)-4- BIS(SUBSTITUTED ARYL) HYDROXYMETHYL]PIPERIDINIUM SALTS

Title (en)

INSECTICIDAL N-(SUBSTITUTED ARYLMETHYL)-4- BIS(SUBSTITUTED ARYL) HYDROXYMETHYL]PIPERIDINIUM SALTS

Title (de)

INSEKTIZIDE [N-(SUBSTITUIERTES ARALMETHYL)-4-BIS(SUBSTITUIERTES ARYL)HYDROXYMETHL] PIPERIDINIUM SALZE

Title (fr)

SELS INSECTICIDES DE N-(ARYLMETHYLE SUBSTITUE)-4- BIS(ARYLE SUBSTITUE)HYDROXYMETHYLE]PIPERIDINIUM

Publication

EP 0912090 A4 (EN)

Application

EP 97931416 A

Priority

  • US 9711077 W
  • US 2113996 P
  • US 85216097 A

Abstract (en)

[origin: WO9800015A1] Compounds of structure (I) are disclosed as effective insecticides, in which Q is hydroxy; U is -(CH2)n-, where n is 1; R is structure (II) in which V, W, Y and Z are each hydrogen; X is alkoxy, cycloalkylalkoxy, alkoxycarbonyl, alkoxycarbonylamino, or a five- or six-membered heteroaryl or heteroaryloxy, each heteroaryl optionally substituted with halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxyalkyl, or haloalkoxyakyl; R<1> and R<2> are independently selected from haloalkyl; phenyl substituted with halogen, halothio, haloalkyl, or haloalkoxy; or a five- or six-membered heteroaryl substituted with halogen or haloalkyl; R<3> is alkyl, haloalkyl, hydroxyalkyl, alkoxyalkyl, dialkylaminoalkyl, alkylaminocarbonyloxyalkyl, alkylthioalkyl, alkylsulfonylalkyl, alkylcarbonyloxalkyl, alkoxycarbonylalkyl, carboxyalkyl, carboxyarylalkyl, arylcarbonyl, sulfonato, or sulfonatoalkyl, and may bear a negative charge resulting in an inner salt; and a separate anion is chloride, bromide, iodide, or a phenyl or alkyl sulfate or sulfonate; with the proviso that at least one of R<1> and R<2> is phenyl substituted in the para position or pyrid-2-yl or pyrimidin-2-yl, each substituted in the 5-position; each aliphatic moiety contains not more than 4 carbon atoms, except that R<3> may contain up to eighteen carbon atoms; halogen means bromine, chlorine, or fluorine; each heteroaryl contains from 1 to 4 nitrogen atoms, or 1 or 2 oxygen or sulfur atoms, or 1 or 2 nitrogen atoms and an oxygen or sulfur atom.

IPC 1-7

A01N 43/08; A01N 43/10; A01N 43/40; A01N 43/54; A01N 55/00; A61K 31/445; A61K 31/505; C07D 211/14; C07D 211/18; C07D 211/20; C07D 239/00

IPC 8 full level

A01N 43/40 (2006.01); A01N 43/54 (2006.01); A01N 43/713 (2006.01); A01N 47/12 (2006.01); C07D 211/14 (2006.01)

CPC (source: EP)

A01N 43/40 (2013.01); A01N 43/54 (2013.01); A01N 43/713 (2013.01); A01N 47/12 (2013.01); C07D 211/14 (2013.01)

Citation (search report)

Designated contracting state (EPC)

DE ES FR GB GR IT

DOCDB simple family (publication)

WO 9800015 A1 19980108; AU 3505197 A 19980121; BR 9710108 A 19990810; EP 0912090 A1 19990506; EP 0912090 A4 20000517

DOCDB simple family (application)

US 9711077 W 19970625; AU 3505197 A 19970625; BR 9710108 A 19970625; EP 97931416 A 19970625