Global Patent Index - EP 0931045 A1

EP 0931045 A1 19990728 - MATRIX METALLOPROTEINASE INHIBITORS AND THEIR THERAPEUTIC USES

Title (en)

MATRIX METALLOPROTEINASE INHIBITORS AND THEIR THERAPEUTIC USES

Title (de)

INHIBITOREN VON MATRIX-METALLPROTEINASEN UND IHRE THERAPEUTISCHE ANWENDUNG

Title (fr)

INHIBITEURS DE METALLOPROTEINASES MATRICIELLES ET LEURS UTILISATIONS PHARMACEUTIQUES

Publication

EP 0931045 A1 19990728 (EN)

Application

EP 97939527 A 19970822

Priority

  • US 9714859 W 19970822
  • US 2506296 P 19960904
  • US 5571397 P 19970807

Abstract (en)

[origin: WO9809934A1] The present invention relates to a method of inhibiting matrix metalloproteinases using compounds that are dibenzofuran sulfonamide derivatives having Formula (I). More particularly, the present invention relates to a method of treating diseases in which matrix metalloproteinases are involved such as multiple sclerosis, atherosclerotic plaque rupture, restenosis, aortic aneurism, heart failure, periodontal disease, corneal ulceration, burns, decubital ulcers, chronic ulcers or wounds, cancer metastasis, tumor angiogenesis, arthritis, or other autoimmune or inflammatory diseases dependent upon tissue invasion by leukocytes.

IPC 1-7

C07C 35/38; C07D 209/82; C07D 333/78; C07D 307/91; A61K 31/195; A61K 31/40; A61K 31/34; A61K 31/38

IPC 8 full level

A61K 31/343 (2006.01); A61K 31/381 (2006.01); A61K 31/403 (2006.01); A61P 1/02 (2006.01); A61P 9/04 (2006.01); A61P 9/10 (2006.01); A61P 17/02 (2006.01); A61P 19/02 (2006.01); A61P 27/02 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07C 311/19 (2006.01); C07D 209/88 (2006.01); C07D 307/91 (2006.01); C07D 333/76 (2006.01)

CPC (source: EP KR)

A61K 31/343 (2013.01 - EP); A61K 31/381 (2013.01 - EP); A61P 1/02 (2017.12 - EP); A61P 9/04 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 17/02 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 27/02 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07C 311/19 (2013.01 - EP); C07D 209/82 (2013.01 - KR); C07D 307/91 (2013.01 - EP); C07D 333/76 (2013.01 - EP); C07C 2603/18 (2017.04 - EP)

Citation (search report)

See references of WO 9809934A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9809934 A1 19980312; AU 4159597 A 19980326; AU 735013 B2 20010628; BR 9711988 A 19990824; CA 2256716 A1 19980312; EP 0931045 A1 19990728; JP 2000517341 A 20001226; KR 20000068414 A 20001125; NZ 333063 A 20001222

DOCDB simple family (application)

US 9714859 W 19970822; AU 4159597 A 19970822; BR 9711988 A 19970822; CA 2256716 A 19970822; EP 97939527 A 19970822; JP 51270998 A 19970822; KR 19997001756 A 19990303; NZ 33306397 A 19970822