EP 0946553 B1 20030129 - 8-AZABICYCLO 3.2.1]OCTANE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INSECTICIDES
Title (en)
8-AZABICYCLO 3.2.1]OCTANE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INSECTICIDES
Title (de)
8-AZABICYCLO 3.2.1]OCTAN-DERIVATE, IHRE HERSTELLUNG UND IHRE VERWENDUNG ALS INSEKTIZIDE
Title (fr)
DERIVES DE 8-AZABICYCLO 3.2.1]OCTANE, LEUR PREPARATION ET LEUR UTILISATION COMME INSECTICIDES
Publication
Application
Priority
- GB 9702986 W 19971030
- GB 9624611 A 19961126
Abstract (en)
[origin: WO9825923A1] A compound of formula (I) wherein Ar is optionally substituted phenyl or optionally substituted 5- or 6-membered heterocyclic ring containing from 1 to 3 heteroatoms individually selected from nitrogen, oxygen and sulfur atoms, and at least one unsaturation (double bond) between adjacent atoms in the ring, said heterocyclic ring being optionally fused to a benzene ring, wherein the substituents, if present, are selected from halogen atoms, cyano, alkyl, alkenyl, alkynyl, alkoxy, haloalkyl, haloalkenyl, alkylthio and alkyl amino groups; R represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkenyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl, dithiocarboxyl or XR<3> (where X represents oxygen or a group NR<4>), provided that when R is alkenyl, aralkenyl or alkynyl said group does not have an unsaturated carbon atom bonding directly to the ring nitrogen of formula (I); R<3> and R<4> are, independently, hydrogen, alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, heterocyclylalkyl, alkoxycarbonyl or carboxylic acyl; alkyl moieties of R, R<3> and R<4> comprise from 1 to 15 carbon atoms, and are optionally substituted with one or more substituents selected from halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, amino, acylamino, imidate and phosphonato groups; aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkanyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl or dithiocarboxyl moieties of R, R<3> and R<4> comprise from 1 to 15 carbon atoms, and are optionally substituted with one or more substituents selected from, halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, haloalkyl, alkyl, amino, acylamino, imidate and phosphonato groups; R<1> represents hydrogen, hydroxy, alkyl, alkoxy, amino, nitro, isocyanato, acylamino, hydroxyalkyl, optionally substituted heteroaryl, alkoxyalkyl, haloalkyl, halohydroxyalkyl, aralkyloxyalkyl, acyloxyalkyl, amidoximido, sulfonyloxyalkyl, aminoalkyl, alkoxycarbonylamino, acylaminoalkyl, cyanoalkyl, imino, formyl, acyl or carboxylic acid or an ester or amide thereof, or alkenyl or alkynyl either of which is optionally substituted by halogen, alkoxy, cycloalkyl, optionally substituted aryl, optionally substituted heteroaryl or cyano; or an acid addition salt, quaternary ammonium salt or <u>N</u>-oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
IPC 1-7
IPC 8 full level
A01N 43/90 (2006.01); A01N 47/16 (2006.01); A01N 47/18 (2006.01); C07D 451/02 (2006.01); C07D 451/04 (2006.01); C07D 451/06 (2006.01); C07D 451/14 (2006.01); C07D 498/08 (2006.01)
CPC (source: EP KR US)
A01N 43/90 (2013.01 - EP US); A01N 47/16 (2013.01 - EP US); A01N 47/18 (2013.01 - EP US); C07D 451/02 (2013.01 - EP KR US); C07D 451/04 (2013.01 - EP US); C07D 451/06 (2013.01 - EP US); C07D 451/14 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE
DOCDB simple family (publication)
WO 9825923 A1 19980618; AT E231860 T1 20030215; AU 4789097 A 19980703; BR 9713429 A 20000201; CA 2272076 A1 19980618; CN 1245498 A 20000223; DE 69718816 D1 20030306; DE 69718816 T2 20031030; EP 0946553 A1 19991006; EP 0946553 B1 20030129; ES 2186876 T3 20030516; GB 9624611 D0 19970115; ID 21772 A 19990722; IL 130059 A0 20000229; JP 2001506988 A 20010529; KR 20000069095 A 20001125; SV 1997000097 A 19981015; TR 199901170 T2 19990721; US 6093726 A 20000725; US 6174894 B1 20010116
DOCDB simple family (application)
GB 9702986 W 19971030; AT 97910543 T 19971030; AU 4789097 A 19971030; BR 9713429 A 19971030; CA 2272076 A 19971030; CN 97181522 A 19971030; DE 69718816 T 19971030; EP 97910543 A 19971030; ES 97910543 T 19971030; GB 9624611 A 19961126; ID 990380 A 19971030; IL 13005997 A 19971030; JP 52633198 A 19971030; KR 19997004558 A 19990524; SV 1997000097 A 19971124; TR 9901170 T 19971030; US 35774999 A 19990721; US 96963997 A 19971113