EP 0954526 A2 19991110 - SERINE PROTEASE INHIBITORS
Title (en)
SERINE PROTEASE INHIBITORS
Title (de)
SUBSTITUIERTE OXADIAZOL, THIADIAZOL UND TRIAZOL SERINPROTEASE INHIBITORE
Title (fr)
INHIBITEURS DE LA SERINE PROTEASE
Publication
Application
Priority
- US 9721636 W 19971205
- US 76119096 A 19961206
- US 76238196 A 19961206
- US 77131796 A 19961206
- US 76091696 A 19961206
- US 76131396 A 19961206
- US 98520197 A 19971204
- US 98488197 A 19971204
- US 98505697 A 19971204
- US 98488497 A 19971204
- US 98529897 A 19971204
Abstract (en)
[origin: WO9824806A2] The present invention relates to certain substituted oxadiazole, thiadiazole and triazole peptoids which are useful as inhibitors of serine proteases.
IPC 1-7
C07K 5/062; C07K 5/078; C07D 413/12; C07D 413/14; C07D 271/10; C07D 417/12
IPC 8 full level
A61K 31/41 (2006.01); A61K 31/4245 (2006.01); A61K 31/433 (2006.01); A61K 31/435 (2006.01); A61K 31/495 (2006.01); A61K 31/513 (2006.01); A61K 38/55 (2006.01); A61K 38/05 (2006.01); A61K 38/06 (2006.01); A61P 43/00 (2006.01); C07D 271/10 (2006.01); C07D 413/12 (2006.01); C07D 413/14 (2006.01); C07D 417/12 (2006.01); C07D 487/02 (2006.01); C07D 491/02 (2006.01); C07D 495/04 (2006.01); C07K 5/02 (2006.01); C07K 5/06 (2006.01); C07K 5/062 (2006.01); C07K 5/065 (2006.01); C07K 5/068 (2006.01); C07K 5/072 (2006.01); C07K 5/078 (2006.01); C07K 5/083 (2006.01); C07K 5/12 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP)
A61P 43/00 (2018.01); C07D 271/10 (2013.01); C07D 413/12 (2013.01); C07D 413/14 (2013.01); C07D 417/12 (2013.01); C07K 5/0202 (2013.01); C07K 5/06026 (2013.01); C07K 5/06043 (2013.01); C07K 5/06052 (2013.01); C07K 5/06078 (2013.01); C07K 5/06086 (2013.01); C07K 5/06104 (2013.01); C07K 5/06139 (2013.01); C07K 5/06156 (2013.01); C07K 5/06191 (2013.01); C07K 5/0806 (2013.01); C07K 5/12 (2013.01); A61K 38/00 (2013.01)
Designated contracting state (EPC)
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9824806 A2 19980611; WO 9824806 A3 19981015; WO 9824806 B1 19990520; AU 5589498 A 19980629; AU 734615 B2 20010621; CA 2272548 A1 19980611; CN 1247542 A 20000315; EP 0954526 A2 19991110; HU P0100669 A2 20010828; HU P0100669 A3 20011228; JP 2001507679 A 20010612; JP 3220169 B2 20011022; NO 992734 D0 19990604; NO 992734 L 19990802; NZ 336046 A 20001027; RU 2217436 C2 20031127; TR 199901681 T2 20000321; TR 200103270 T2 20030321
DOCDB simple family (application)
US 9721636 W 19971205; AU 5589498 A 19971205; CA 2272548 A 19971205; CN 97180392 A 19971205; EP 97952232 A 19971205; HU P0100669 A 19971205; JP 52565698 A 19971205; NO 992734 A 19990604; NZ 33604697 A 19971205; RU 99114606 A 19971205; TR 200103270 T 19971205; TR 9901681 T 19971205