EP 0969840 A1 20000112 - THROMBIN INHIBITORS
Title (en)
THROMBIN INHIBITORS
Title (de)
THROMBIN INHIBITOREN
Title (fr)
INHIBITEURS DE THROMBINE
Publication
Application
Priority
- GB 9716872 A 19970808
- GB 9800214 A 19980106
- US 9805486 W 19980320
- US 4154397 P 19970324
- US 4756197 P 19970522
Abstract (en)
[origin: WO9842342A1] A compound which inhibits human thrombin and has structure (I) or (II) or (III) and pharmaceutically acceptable salts thereof, wherein compounds such as (IV) are useful for inhibiting formation of blood platelet aggregates in blood in a mammal.
IPC 1-7
A61K 31/495; A61K 31/535; C07D 401/14; C07D 403/12; C07D 413/06
IPC 8 full level
A61K 31/427 (2006.01); A61K 31/4439 (2006.01); A61K 31/454 (2006.01); A61K 31/4545 (2006.01); A61K 31/497 (2006.01); A61K 31/5377 (2006.01); A61K 38/00 (2006.01); A61P 7/02 (2006.01); A61P 43/00 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 403/12 (2006.01); C07D 403/14 (2006.01); C07D 405/14 (2006.01); C07D 417/12 (2006.01); C07K 5/00 (2006.01); C07K 5/02 (2006.01); C07K 5/078 (2006.01)
CPC (source: EP)
A61P 7/02 (2017.12); A61P 43/00 (2017.12); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 403/12 (2013.01); C07K 5/0207 (2013.01); C07K 5/06139 (2013.01); A61K 38/00 (2013.01)
Designated contracting state (EPC)
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9842342 A1 19981001; AU 6572798 A 19981020; AU 728006 B2 20010104; CA 2283704 A1 19981001; EP 0969840 A1 20000112; EP 0969840 A4 20010228; JP 2001518932 A 20011016
DOCDB simple family (application)
US 9805486 W 19980320; AU 6572798 A 19980320; CA 2283704 A 19980320; EP 98911875 A 19980320; JP 54582598 A 19980320