Global Patent Index - EP 0969840 A4

EP 0969840 A4 20010228 - THROMBIN INHIBITORS

Title (en)

THROMBIN INHIBITORS

Title (de)

THROMBIN INHIBITOREN

Title (fr)

INHIBITEURS DE THROMBINE

Publication

EP 0969840 A4 20010228 (EN)

Application

EP 98911875 A 19980320

Priority

  • GB 9716872 A 19970808
  • GB 9800214 A 19980106
  • US 9805486 W 19980320
  • US 4154397 P 19970324
  • US 4756197 P 19970522

Abstract (en)

[origin: WO9842342A1] A compound which inhibits human thrombin and has structure (I) or (II) or (III) and pharmaceutically acceptable salts thereof, wherein compounds such as (IV) are useful for inhibiting formation of blood platelet aggregates in blood in a mammal.

IPC 1-7

A61K 31/495; A61K 31/535; C07D 401/14; C07D 403/12; C07D 413/06; C07D 401/12; C07K 5/06

IPC 8 full level

A61K 31/427 (2006.01); A61K 31/4439 (2006.01); A61K 31/454 (2006.01); A61K 31/4545 (2006.01); A61K 31/497 (2006.01); A61K 31/5377 (2006.01); A61K 38/00 (2006.01); A61P 7/02 (2006.01); A61P 43/00 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 403/12 (2006.01); C07D 403/14 (2006.01); C07D 405/14 (2006.01); C07D 417/12 (2006.01); C07K 5/00 (2006.01); C07K 5/02 (2006.01); C07K 5/078 (2006.01)

CPC (source: EP)

A61P 7/02 (2017.12); A61P 43/00 (2017.12); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 403/12 (2013.01); C07K 5/0207 (2013.01); C07K 5/06139 (2013.01); A61K 38/00 (2013.01)

Citation (search report)

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9842342 A1 19981001; AU 6572798 A 19981020; AU 728006 B2 20010104; CA 2283704 A1 19981001; EP 0969840 A1 20000112; EP 0969840 A4 20010228; JP 2001518932 A 20011016

DOCDB simple family (application)

US 9805486 W 19980320; AU 6572798 A 19980320; CA 2283704 A 19980320; EP 98911875 A 19980320; JP 54582598 A 19980320