EP 0975629 A1 20000202 - TREATMENT OR PROPHYLAXIS OF PROSTATIC CANCER AND BENIGN PROSTATIC HYPERPLASIA WITH SELECTIVE ESTROGEN RECEPTOR MODULATORS
Title (en)
TREATMENT OR PROPHYLAXIS OF PROSTATIC CANCER AND BENIGN PROSTATIC HYPERPLASIA WITH SELECTIVE ESTROGEN RECEPTOR MODULATORS
Title (de)
BEHANDLUNG ODER PROPHYLAXE VON PROSTATAKREBS UND DER GUTARTIGEN PROSTATEHYPERPLASIEMIT SELEKTIVEN ÖSTROGENREZEPTOR-MODULATOREN
Title (fr)
TRAITEMENT OU PROPHYLAXIE DU CANCER DE LA PROSTATE ET DE L'HYPERPLASIE PROSTATIQUE BENIGNE A L'AIDE DE MODULATEURS SELECTIFS DES RECEPTEURS D'OESTROGENES
Publication
Application
Priority
- US 9807274 W 19980407
- US 4322397 P 19970409
Abstract (en)
[origin: WO9845288A1] The present invention provides a method for the treatment or prophylaxis of benign prostatic hyperplasia or prostatic cancer in a patient in need of such treatment comprising administering a selective estrogen receptor modulating compound of formula (I), in which R<1> and R<2> are independently hydroxy and alkoxy of one to four carbon atoms; and R<3> and R<4> are independently methyl or ethyl, or R<3> and R<4>, taken together with the nitrogen atom to which they are attached, form a pyrrolidino, methyl-pyrrolidino, dimethylpyrrolidino, piperidino, morpholino, or hexamethyleneimino ring.
IPC 1-7
IPC 8 full level
A61K 31/381 (2006.01); A61K 31/4025 (2006.01); A61K 31/4535 (2006.01); A61K 31/5377 (2006.01); A61K 31/55 (2006.01); A61P 5/30 (2006.01); A61P 13/00 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 333/64 (2006.01)
CPC (source: EP KR)
A61K 31/38 (2013.01 - KR); A61K 31/381 (2013.01 - EP); A61K 31/4025 (2013.01 - EP); A61K 31/4535 (2013.01 - EP); A61K 31/5377 (2013.01 - EP); A61K 31/55 (2013.01 - EP); A61P 5/30 (2017.12 - EP); A61P 13/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE
DOCDB simple family (publication)
WO 9845288 A1 19981015; AU 6966198 A 19981030; BR 9808515 A 20010619; CA 2286204 A1 19981015; CN 1259944 A 20000712; EA 199900914 A1 20000424; EP 0975629 A1 20000202; EP 0975629 A4 20010321; HU 0003589 A2 20020128; HU 0003589 A3 20020228; ID 24358 A 20000713; IL 132277 A0 20010319; JP 2001518900 A 20011016; KR 20010006218 A 20010126; NO 994903 D0 19991008; NO 994903 L 19991209; PL 336205 A1 20000605; TR 199902701 T2 20000221; ZA 982819 B 19991004
DOCDB simple family (application)
US 9807274 W 19980407; AU 6966198 A 19980407; BR 9808515 A 19980407; CA 2286204 A 19980407; CN 98805956 A 19980407; EA 199900914 A 19980407; EP 98915488 A 19980407; HU 0003589 A 19980407; ID 991188 A 19980407; IL 13227798 A 19980407; JP 54316898 A 19980407; KR 19997009298 A 19991009; NO 994903 A 19991008; PL 33620598 A 19980407; TR 9902701 T 19980407; ZA 982819 A 19980402