EP 0975633 A1 20000202 - 5,6,7-TRISUBSTITUTED-4-AMINOPYRIDOL 2,3-D PYRIMIDINE COMPOUNDS
Title (en)
5,6,7-TRISUBSTITUTED-4-AMINOPYRIDOL 2,3-D PYRIMIDINE COMPOUNDS
Title (de)
5,6,7-TRISUBSTITUIERTE-4-AMINOPYRIDO(2,3-D)PYRIMIDIN VERBINDUNGEN
Title (fr)
COMPOSES DE 4-AMINOPYRIDOL 2,3-D PYRIMIDINE A TRISUBSTITUTION 5,6,7
Publication
Application
Priority
- US 9807201 W 19980413
- US 84348497 A 19970416
Abstract (en)
[origin: WO9846604A1] A compound having formula (II) wherein R<1>, R<2>, R<3>, R<4> and R<5> are defined, a method for inhibiting adenosine kinase by administering a compound thereof, a pharmaceutical composition comprising a therapeutically effective amount of a compound thereof above in combination with a pharmaceutically acceptable carrier, a method of treating cerebral ischemia, epilepsy, pain, nociperception, inflammation and sepsis in a mammal in need of such treatment, comprising administering to the mammal a therapeutically effective amount of a compound thereof, and methods for preparation thereof.
IPC 1-7
IPC 8 full level
A61K 31/519 (2006.01); A61P 1/00 (2006.01); A61P 25/04 (2006.01); A61P 3/10 (2006.01); A61P 9/00 (2006.01); A61P 25/08 (2006.01); A61P 25/18 (2006.01); A61P 25/22 (2006.01); A61P 29/00 (2006.01); A61P 31/00 (2006.01); A61P 37/06 (2006.01); A61P 43/00 (2006.01); C07D 471/04 (2006.01)
CPC (source: EP KR)
A61P 1/00 (2018.01 - EP); A61P 3/10 (2018.01 - EP); A61P 9/00 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 19/02 (2018.01 - EP); A61P 25/04 (2018.01 - EP); A61P 25/08 (2018.01 - EP); A61P 25/18 (2018.01 - EP); A61P 25/22 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 31/00 (2018.01 - EP); A61P 37/06 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07D 471/04 (2013.01 - EP KR)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE
Designated extension state (EPC)
RO SI
DOCDB simple family (publication)
WO 9846604 A1 19981022; AR 012437 A1 20001018; AU 7108098 A 19981111; AU 741033 B2 20011122; BG 103853 A 20000630; BR 9809056 A 20000801; CA 2286592 A1 19981022; CN 1252069 A 20000503; CO 4940470 A1 20000724; EP 0975633 A1 20000202; HU P0001443 A2 20001028; HU P0001443 A3 20010129; IL 131617 A0 20010128; JP 2001520654 A 20011030; KR 20010006462 A 20010126; NO 995035 D0 19991015; NO 995035 L 19991215; NZ 337125 A 20010629; PL 336265 A1 20000619; SK 140099 A3 20000516; TR 199902550 T2 20000421; ZA 983175 B 19981021
DOCDB simple family (application)
US 9807201 W 19980413; AR P980101734 A 19980415; AU 7108098 A 19980413; BG 10385399 A 19991103; BR 9809056 A 19980413; CA 2286592 A 19980413; CN 98804117 A 19980413; CO 98020978 A 19980416; EP 98918091 A 19980413; HU P0001443 A 19980413; IL 13161798 A 19980413; JP 54408398 A 19980413; KR 19997009552 A 19991015; NO 995035 A 19991015; NZ 33712598 A 19980413; PL 33626598 A 19980413; SK 140099 A 19980413; TR 9902550 T 19980413; ZA 983175 A 19980415