Global Patent Index - EP 0986549 A1

EP 0986549 A1 20000322 - DESOXYCYCLODEPSIPEPTIDES AND THEIR USE FOR COMBATTING ENDOPARASITES

Title (en)

DESOXYCYCLODEPSIPEPTIDES AND THEIR USE FOR COMBATTING ENDOPARASITES

Title (de)

DESOXYCYCLODEPSIPEPTIDE UND IHRE VERWENDUNG ZUR BEKÄMPFUNG VON ENDOPARASITEN

Title (fr)

DESOXYCYCLODEPSIPEPTIDES ET LEUR UTILISATION POUR LA LUTTE CONTRE LES ENDOPARASITES

Publication

EP 0986549 A1 20000322 (DE)

Application

EP 98930724 A 19980525

Priority

  • DE 19723320 A 19970604
  • DE 19810017 A 19980309
  • EP 9803059 W 19980525

Abstract (en)

[origin: WO9855469A1] The invention relates to novel desoxycyclodepsipeptides of formula (I) in which C=X<1>, C=X<2>, C=X<3> and C=X<4> independently of each other respectively represent one of the CO, CS or CH2 groups, with at least one of these groups representing CH2. The invention also relates to their mixtures and derivatives. Said compounds are produced from cyclodepsipeptides having 24 ring members formed by alternating alpha -amino carboxylic acids and alpha -hydroxy carboxylic acids by complete or partial chemoselective reduction of the carbonyl groups of the amide function into methylene groups, using suitable reduction methods. The desoxycyclodepsipeptides produced according to the invention have an anthelmintic effect.

IPC 1-7

C07D 273/00; C07D 413/14; C07D 413/10; A61K 31/395

IPC 8 full level

A61K 31/341 (2006.01); A61K 31/395 (2006.01); A61K 31/4025 (2006.01); A61K 31/4035 (2006.01); A61K 31/496 (2006.01); A61K 31/5377 (2006.01); A61K 31/55 (2006.01); A61P 33/00 (2006.01); A61P 33/10 (2006.01); C07D 273/00 (2006.01); C07D 413/10 (2006.01); C07D 413/14 (2006.01)

CPC (source: EP US)

A61P 33/00 (2017.12 - EP); A61P 33/10 (2017.12 - EP); C07D 273/00 (2013.01 - EP US); C07D 413/10 (2013.01 - EP US); C07D 413/14 (2013.01 - EP US)

Citation (search report)

See references of WO 9855469A1

Designated contracting state (EPC)

AT BE CH DE DK ES FR GB IT LI NL

DOCDB simple family (publication)

WO 9855469 A1 19981210; AU 735424 B2 20010705; AU 8105998 A 19981221; BR 9810412 A 20000822; CA 2292698 A1 19981210; CN 1076349 C 20011219; CN 1259129 A 20000705; EP 0986549 A1 20000322; HK 1028605 A1 20010223; JP 2002502398 A 20020122; NZ 501478 A 20010525; US 6355615 B1 20020312

DOCDB simple family (application)

EP 9803059 W 19980525; AU 8105998 A 19980525; BR 9810412 A 19980525; CA 2292698 A 19980525; CN 98805881 A 19980525; EP 98930724 A 19980525; HK 00108014 A 20001213; JP 50141599 A 19980525; NZ 50147898 A 19980525; US 42480399 A 19991129