Global Patent Index - EP 0991639 A1

EP 0991639 A1 20000412 - 4- (1H-IMIDAZOL-4-YL)PIPERIDIN-1-YL ANILIDE DERIVATIVES, THEIR PREPARATION AND APPLICATION IN THERAPY

Title (en)

4- (1H-IMIDAZOL-4-YL)PIPERIDIN-1-YL ANILIDE DERIVATIVES, THEIR PREPARATION AND APPLICATION IN THERAPY

Title (de)

4-¬(1H-IMIDAZOL-4-YL)PIPERIDIN-1-YL ANILID DERIVATE, IHRE HERSTELLUNG UND VERWENDUNG ALS ARZNEIMITTEL

Title (fr)

DERIVES DE 4- (1H-IMIDAZOL-4-YL)PIPERIDIN-1-YL ANILIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE

Publication

EP 0991639 A1 20000412 (FR)

Application

EP 98932237 A 19980619

Priority

  • FR 9801288 W 19980619
  • FR 9707900 A 19970625

Abstract (en)

[origin: FR2765221A1] The invention concerns compounds of formula (I) in which R1 represents a hydrogen atom or a linear or branched (C1-C4) alkyl group; R2 represents a linear or branched (C1-C6) alkyl, cyclo(C3-C7) alkyl or cyclo(C3-C7)alkyl(C1-C5) alkyl group; R3 represents a -OR4, -O(CH2)nNR5R6, -NHC(NH)NH2, -NHC(NH)N(CH3)2, -NR5R6, -NR5(CH2)nNR6R7 group, a group (a), X being selected among the oxygen and sulphur atoms and the -CHR8, -NR8, -SO- and -SO2- groups; R4, R5, R6, R7 and R8 being a hydrogen atom, a linear or branched (C1-C6)alkyl, cyclo (C3-C7)alkyl, cyclo(C3-C7)alkyl(C1-C5)alkyl, phenyl, phenyl(C1-C6)alkyl or heteroaryl group; m = 1 or 2 and n = 2, 3 or 4. The invention is applicable in therapy.

IPC 1-7

C07D 401/04; A61K 31/415; C07D 401/14

IPC 8 full level

A61K 31/454 (2006.01); A61K 31/496 (2006.01); A61K 31/5377 (2006.01); A61K 31/551 (2006.01); A61P 9/00 (2006.01); A61P 43/00 (2006.01); C07D 401/04 (2006.01); C07D 401/14 (2006.01)

CPC (source: EP)

A61P 9/00 (2017.12); A61P 43/00 (2017.12); C07D 401/04 (2013.01); C07D 401/14 (2013.01)

Citation (search report)

See references of WO 9900379A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

Designated extension state (EPC)

AL LT LV MK RO SI

DOCDB simple family (publication)

FR 2765221 A1 19981231; FR 2765221 B1 19990730; AR 013127 A1 20001213; AU 8220698 A 19990119; EP 0991639 A1 20000412; JP 2002506458 A 20020226; WO 9900379 A1 19990107; ZA 985518 B 19990128

DOCDB simple family (application)

FR 9707900 A 19970625; AR P980103032 A 19980624; AU 8220698 A 19980619; EP 98932237 A 19980619; FR 9801288 W 19980619; JP 50531399 A 19980619; ZA 985518 A 19980624