Global Patent Index - EP 1000026 A1

EP 1000026 A1 20000517 - SPECIAL 3-AZABICYCLO 3.1.0 HEXANES, METHOD FOR PRODUCING AND MODIFYING THE SAME, AND THEIR USE

Title (en)

SPECIAL 3-AZABICYCLO 3.1.0 HEXANES, METHOD FOR PRODUCING AND MODIFYING THE SAME, AND THEIR USE

Title (de)

SPEZIELLE 3-AZABICYCLO 3.1.0 HEXANE, VERFAHREN ZU DEREN HERSTELLUNG UND MODIFIZIERUNG SOWIE DEREN VERWENDUNG

Title (fr)

3-AZABICYCLO 3.1.0 HEXANES SPECIAUX, LEUR PROCEDE DE PREPARATION ET DE MODIFICATION, AINSI QUE LEUR UTILISATION

Publication

EP 1000026 A1 20000517 (DE)

Application

EP 98937579 A 19980721

Priority

  • DE 19733439 A 19970802
  • EP 9804542 W 19980721

Abstract (en)

[origin: WO9906368A1] The invention relates to novel 3-azabicyclo[3.1.0]hexanes with a doubly protected amino group in position 6, and to a method for producing the same from chloramines or bicyclic N,O acetals or bicyclic nitriles. The two protective groups on the amino group in 6 and the group on N(3) can be specifically removed. The novel 3-azabicyclo[3.1.0]hexanes with a doubly protected amino group in position 6 are suitable for manufacturing pharmaceutical products, e.g. gyrase inhibitors, which can be modified by subsequently splitting off the protective groups.

IPC 1-7

C07D 209/52; A61K 31/47; C07D 471/04

IPC 8 full level

A61K 31/4375 (2006.01); A61K 31/47 (2006.01); C07D 209/52 (2006.01); C07D 471/14 (2006.01); C07D 471/04 (2006.01)

CPC (source: EP US)

C07D 209/52 (2013.01 - EP US); C07D 471/14 (2013.01 - EP US); Y02P 20/55 (2015.11 - EP US)

Designated contracting state (EPC)

BE CH DE ES FI FR GB IE IT LI NL PT SE

DOCDB simple family (publication)

WO 9906368 A1 19990211; AU 8632198 A 19990222; CA 2298509 A1 19990211; CN 1265650 A 20000906; DE 19733439 A1 19990204; EP 1000026 A1 20000517; HU P0002895 A2 20010228; HU P0002895 A3 20010428; IL 134058 A0 20010430; JP 2001512101 A 20010821; KR 20010022512 A 20010315; PL 338349 A1 20001023; US 6310216 B1 20011030

DOCDB simple family (application)

EP 9804542 W 19980721; AU 8632198 A 19980721; CA 2298509 A 19980721; CN 98807850 A 19980721; DE 19733439 A 19970802; EP 98937579 A 19980721; HU P0002895 A 19980721; IL 13405898 A 19980721; JP 2000505127 A 19980721; KR 20007001100 A 20000201; PL 33834998 A 19980721; US 46386700 A 20000218