Global Patent Index - EP 1000030 A1

EP 1000030 A1 2000-05-17 - PIPERIDINE OLIGOMERS AND COMBINATORIAL LIBRARIES THEREOF

Title (en)

PIPERIDINE OLIGOMERS AND COMBINATORIAL LIBRARIES THEREOF

Title (de)

PIPERIDIN-OLIGOMEREN UND DIESE ENTHALTENDE KOMBINATORISCHE BIBLIOTHEKEN

Title (fr)

OLIGOMERES DE PIPERIDINE ET BANQUES COMBINATOIRES DE CEUX-CI

Publication

EP 1000030 A1 (EN)

Application

EP 98933574 A

Priority

  • DK 9800330 W
  • DK 85897 A

Abstract (en)

[origin: WO9903832A1] The present invention relates to piperidine oligomers, methods for the preparation of piperidine oligomers and compound libraries thereof, and the use of piperidine oligomers as drug substances. The present invention also relates to the use of combinatorial libraries of piperidine oligomers for screening purposes. The oligomers have one of the general formulas (I) or (II). Each of the monomers (piperidine carboxylic acids) are linked via amide bonds. The piperidine monomers may carry substituents, particularly hydroxy, hydroxymethyl, and carboxy substituents. The oligomers may be prepared in libraries (arrays) of compounds especially suitable for screening purposes.

IPC 1-7 (main, further and additional classification)

C07D 211/62; A61K 31/445; C07D 471/22

IPC 8 full level (invention and additional information)

C07D 211/62 (2006.01); C07D 471/22 (2006.01); C07B 61/00 (2006.01)

CPC (invention and additional information)

C07D 211/62 (2013.01); C40B 40/00 (2013.01)

Citation (search report)

See references of WO 9903832A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

EPO simple patent family

WO 9903832 A1 19990128; AU 8334498 A 19990210; CA 2296428 A1 19990128; EP 1000030 A1 20000517

INPADOC legal status


2001-07-25 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20010201

2000-07-05 [D17P] REQUEST FOR EXAMINATION FILED (DELETED)

2000-05-17 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20000214

2000-05-17 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE