Global Patent Index - EP 1001947 A1

EP 1001947 A1 20000524 - PROCESS FOR MANUFACTURING FLUCONAZOLE

Title (en)

PROCESS FOR MANUFACTURING FLUCONAZOLE

Title (de)

VERFAHREN ZUR HERSTELLUNG VON FLUCONAZOL

Title (fr)

PROCEDE DE FABRICATION DE FLUCONAZOLE

Publication

EP 1001947 A1 20000524 (EN)

Application

EP 98902274 A 19980124

Priority

  • KR 9800018 W 19980124
  • KR 19970002700 A 19970129

Abstract (en)

[origin: WO9832744A1] The invention herein relates to a process for the manufacture of fluconazole, or more particularly, to the process for the manufacture of fluconazole of Formula (1) having superior antifungal activity with a high yield and purity, and its pharmaceutically acceptable salt or hydrate, wherein one-pot reaction is utilized under the mild reaction condition and short reaction time by means of using three compounds expressed by formulae (2, 3 and 4), respectively, in the presence of a base.

IPC 1-7

C07D 249/08

IPC 8 full level

C07D 249/08 (2006.01); C07D 521/00 (2006.01)

CPC (source: EP KR)

C07D 231/12 (2013.01 - EP); C07D 233/56 (2013.01 - EP); C07D 249/08 (2013.01 - EP KR); C07D 403/06 (2013.01 - KR)

Designated contracting state (EPC)

FR

DOCDB simple family (publication)

WO 9832744 A1 19980730; AU 5882398 A 19980818; CZ 308398 A3 19990317; EP 1001947 A1 20000524; HU P0000726 A2 20001128; HU P0000726 A3 20020228; KR 100194945 B1 19990615; KR 19980066917 A 19981015; PL 329117 A1 19990315; SK 133298 A3 19990413

DOCDB simple family (application)

KR 9800018 W 19980124; AU 5882398 A 19980124; CZ 308398 A 19980124; EP 98902274 A 19980124; HU P0000726 A 19980124; KR 19970002700 A 19970129; PL 32911798 A 19980124; SK 133298 A 19980124