Global Patent Index - EP 1005461 A1

EP 1005461 A1 2000-06-07 - ACYLATED 5-AMINOISOTHIAZOLES AS PESTICIDES AND FUNGICIDES

Title (en)

ACYLATED 5-AMINOISOTHIAZOLES AS PESTICIDES AND FUNGICIDES

Title (de)

ACYLIERTE 5-AMINOISOTHIAZOLE ALS PESTIZIDE UND FUNGIZIDE

Title (fr)

5-AMINOISOTHIAZOLES ACYLES A USAGE DE PESTICIDES ET DE FUNGICIDES

Publication

EP 1005461 A1 (DE)

Application

EP 98945190 A

Priority

  • DE 19736545 A
  • EP 9805045 W

Abstract (en)

[origin: DE19736545A1] Acylated 5-aminoisothiazole derivatives (I) are new. Acylated 5-aminoisothiazole derivatives of formula (I) are new. R1 = alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, alkoxy, alkylthio, alkylamino, dialkylamino or optionally substituted cycloalkyl; R2 = H, halo, CN, NO2, thiocyanato, alkoxycarbonyl, alkenyloxycarbonyl, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, thiocarbamoyl, alkoxy, formyl, alkylcarbonyl or CR7=NOR8; R7, R8 = H, alkyl, haloalkyl, alkenyl, optionally substituted cycloalkyl or cycloalkylalkyl or optionally substituted aryl or arylalkyl; R3 = alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, alkenyl, alkynyl, alkylcarbonyloxyalkyl, alkoxycarbonyloxyalkyl, optionally substituted aryl, aralkyl or arylalkoxyalkyl, optionally substituted cycloalkyl, cycloalkylalkyl, cycloalkoxyalkyl or cycloalkylthioalkyl or N=CR5R6; R5, R6 = H, alkyl, haloalkyl, alkenyl, optionally substituted cycloalkyl or cycloalkylalkyl or optionally substituted aryl or arylalkyl; or R5+R6 = an optionally substituted carbocyclic ring; R4 = optionally substituted aryl, cycloalkyl, cycloalkenyl or heterocyclyl; A, Z = O or S; Y = optionally substituted alkylene, alkenylene or alkyleneoxy. Independent claims are included for the following: (a) the preparation of (I); and (b) intermediates of formula (IV) and (VIA). R21 = R, CO-R71 or CR71=NOR7; R = alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, akylsulfonyl or haloalkylsulfonyl; R71 = H or alkyl; R8 = H, 1-4C alkyl, 1-4C haloalkyl, 2-4C alkenyl, 3-6C cycloalkyl or 3-6C cycloalkyl-(1-4C alkyl) (both optionally substituted by 1-3 from 1-4C alkyl or halo groups) or phenyl or phenyl-(1-4C alkyl) (both optionally ring-substituted by 1-3 from halo, NO2, CN, 1-4C alkyl, 1- or 2C haloalkyl, 1-4C alkoxy, 1-4C alkylthio, 1- or 2C haloalkoxy or 1- or 2C haloalkylthio groups) or (1-4C alkoxy)carbonyl or (1-4C alkyl)carbonyloxy.

IPC 1-7 (main, further and additional classification)

C07D 275/03; A01N 43/80

IPC 8 full level (invention and additional information)

C07D 275/02 (2006.01); A01N 43/80 (2006.01); A01N 47/18 (2006.01); C07D 275/03 (2006.01)

CPC (invention and additional information)

C07D 275/03 (2013.01); A01N 47/18 (2013.01)

Citation (search report)

See references of WO 9910334A1

Designated contracting state (EPC)

AT BE CH DE ES FR GB IT LI NL

EPO simple patent family

DE 19736545 A1 19990225; AR 015152 A1 20010418; AU 9259498 A 19990316; EP 1005461 A1 20000607; JP 2001514175 A 20010911; WO 9910334 A1 19990304; ZA 9807585 B 19990223

INPADOC legal status


2002-10-16 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20020301

2000-06-07 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20000322

2000-06-07 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH DE ES FR GB IT LI NL