Global Patent Index - EP 1007042 A1

EP 1007042 A1 20000614 - NOVEL HETEROARYL COMPOUNDS FOR THE MODULATION OF PROTEIN TYROSINE ENZYME RELATED CELLULAR SIGNAL TRANSDUCTION

Title (en)

NOVEL HETEROARYL COMPOUNDS FOR THE MODULATION OF PROTEIN TYROSINE ENZYME RELATED CELLULAR SIGNAL TRANSDUCTION

Title (de)

NEUE HETEROZYKLISCHE VERBINDUNGEN ZUR MODULATION DER PROTEIN-TYROSIN-ENZYM-VERWANDTEN ZELLULÄREN SIGNALTRANSDUKTION

Title (fr)

NOUVEAUX COMPOSES HETEROARYLE POUR LA MODULATION DE LA TRANSDUCTION DE SIGNAUX CELLULAIRES ASSOCIEE AUX ENZYMES PROTEINE TYROSINE

Publication

EP 1007042 A1 20000614 (EN)

Application

EP 98929059 A 19980612

Priority

  • US 9812333 W 19980612
  • US 4956097 P 19970613

Abstract (en)

[origin: WO9856376A1] The present invention relates to novel heteroaryl compounds and the physiologically acceptable salts and the prodrugs thereof which are expected to modulate the activity of protein tyrosine enzymes which are related to cellular signal transduction, in particular, protein tyrosine phosphatase, and therefore are expected to be useful in the prevention and treatment of disorders associated with abnormal protein tyrosine enzyme related cellular signal transduction such as cancer and diabetes.

IPC 1-7

A61K 31/44; A61K 31/47; A61K 31/53; A61K 31/54; A61K 31/425; A61K 31/445; A61K 31/495; A61K 31/505; A61K 31/535; C07D 215/02; C07D 237/26; C07D 239/02; C07D 241/36; C07D 249/02; C07D 251/72; C07D 253/10; C07D 261/20

IPC 8 full level

A61K 31/41 (2006.01); A61K 31/4178 (2006.01); A61K 31/4196 (2006.01); A61K 31/422 (2006.01); A61K 31/424 (2006.01); A61K 31/427 (2006.01); A61K 31/428 (2006.01); A61K 31/433 (2006.01); A61K 31/4436 (2006.01); A61K 31/4439 (2006.01); A61K 31/497 (2006.01); A61K 31/501 (2006.01); A61K 31/506 (2006.01); A61K 31/519 (2006.01); A61K 31/52 (2006.01); A61K 31/522 (2006.01); A61K 31/53 (2006.01); A61K 31/5377 (2006.01); A61K 31/54 (2006.01); A61K 31/55 (2006.01); A61P 3/10 (2006.01); A61P 9/00 (2006.01); A61P 19/02 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 277/20 (2006.01); C07D 277/58 (2006.01); C07D 277/70 (2006.01); C07D 403/06 (2006.01); C07D 409/12 (2006.01); C07D 409/14 (2006.01); C07D 413/14 (2006.01); C07D 417/12 (2006.01); C07D 417/14 (2006.01); C07D 471/04 (2006.01); C07D 473/08 (2006.01); C07D 473/24 (2006.01); C07D 475/02 (2006.01); C07D 487/04 (2006.01); C07D 498/04 (2006.01)

CPC (source: EP)

A61P 3/10 (2017.12); A61P 9/00 (2017.12); A61P 19/02 (2017.12); A61P 29/00 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 409/12 (2013.01); C07D 417/12 (2013.01); C07D 417/14 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 9856376 A1 19981217; AU 8071698 A 19981230; CA 2293400 A1 19981217; EP 1007042 A1 20000614; EP 1007042 A4 20010704; JP 2002512628 A 20020423

DOCDB simple family (application)

US 9812333 W 19980612; AU 8071698 A 19980612; CA 2293400 A 19980612; EP 98929059 A 19980612; JP 50329999 A 19980612