EP 1007073 A1 20000614 - METHODS OF MODIFYING FEEDING BEHAVIOR, COMPOUNDS USEFUL IN SUCH METHODS, AND DNA ENCODING A HYPOTHALAMIC ATYPICAL NEUROPEPTIDE Y/PEPTIDE YY RECEPTOR (Y5)
Title (en)
METHODS OF MODIFYING FEEDING BEHAVIOR, COMPOUNDS USEFUL IN SUCH METHODS, AND DNA ENCODING A HYPOTHALAMIC ATYPICAL NEUROPEPTIDE Y/PEPTIDE YY RECEPTOR (Y5)
Title (de)
VERFAHREN ZUR ÄNDERUNG DER ESSGEWOHNHEITEN, FÜR DIESE VERFAHREN GEEIGNETE VERBINDUNGEN, SOWIE EINE FÜR EINEN HYPOTHALAMISCHES ATYPISCHES NEUROPEPTID Y/ PEPTIDE YY REZEPTOR KODIERENDE DNA
Title (fr)
PROCEDES DE MODIFICATION DU COMPORTEMENT ALIMENTAIRE, COMPOSES UTILES DANS LESDITS PROCEDES, ET ADN CODANT UN RECEPTEUR Y5 ATYPIQUE HYPOTHALAMIQUE DE NEUROPEPTIDE Y/PEPTIDE YY
Publication
Application
Priority
- US 9709504 W 19970604
- US 66865096 A 19960604
- US 80360097 A 19970221
Abstract (en)
[origin: WO9746250A1] The invention provides methods of modifying feeding behavior, including increasing or decreasing food consumption, e.g., in connection with treating obesity, bulimia or anorexia. These methods involve administration of compounds that are selective agonists or antagonists for the Y5 receptor. One such compound has structure (I). In addition, this invention provides an isolated nucleic acid molecule encoding a Y5 receptor, an isolated Y5 receptor protein, vectors comprising an isolated nucleic acid molecule encoding a Y5 receptor, cells comprising such vectors, antibodies directed to the Y5 receptor, nucleic acid probes useful for detecting nucleic acid encoding Y5 receptors, antisense aligonucleotides complementary to any unique sequences of a nucleic acid molecule which encodes a Y5 receptor, and nonhuman transgenic animals which express DNA encoding a normal or a mutant Y5 receptor.
IPC 1-7
A61K 38/02; A61K 39/395; A61K 48/00; C07H 21/02; C07H 21/04; C07K 14/00; C07K 14/435; C07K 14/705; C07K 16/00; C12N 15/00; C12N 15/12
IPC 8 full level
C07K 14/705 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP)
C07K 14/70571 (2013.01); A01K 2217/05 (2013.01); A61K 38/00 (2013.01)
Designated contracting state (EPC)
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 9746250 A1 19971211; AU 3295297 A 19980105; EP 1007073 A1 20000614; EP 1007073 A4 20020327
DOCDB simple family (application)
US 9709504 W 19970604; AU 3295297 A 19970604; EP 97928786 A 19970604