Global Patent Index - EP 1011667 A4

EP 1011667 A4 20010328 - ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (en)

ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (de)

ANTAGONISTEN DES GONADOTROPHIN FREISETZUNGS HORMONS

Title (fr)

ANTAGONISTES DE L'HORMONE DE LIBERATION DE LA GONADOTROPHINE

Publication

EP 1011667 A4 20010328 (EN)

Application

EP 98926171 A 19980601

Priority

  • GB 9719839 A 19970918
  • GB 9800451 A 19980109
  • US 9811204 W 19980601
  • US 4863797 P 19970605
  • US 4863697 P 19970605

Abstract (en)

[origin: WO9855119A1] There are disclosed compounds of formula (I) and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men and women.

IPC 1-7

A61K 31/41; A61K 31/44; C07D 249/08; C07D 257/04; C07D 271/06; C07D 401/14; C07D 403/12; C07D 413/12; C07D 521/00; C07D 487/08; C07D 401/12; C07D 471/08; A61K 38/09; A61P 5/02

IPC 8 full level

A61K 31/41 (2006.01); A61K 31/4196 (2006.01); A61K 31/4439 (2006.01); A61K 38/09 (2006.01); A61K 38/22 (2006.01); A61K 45/00 (2006.01); A61P 5/24 (2006.01); A61P 13/08 (2006.01); A61P 15/00 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 249/08 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01); C07D 413/12 (2006.01); C07D 471/08 (2006.01); C07D 487/08 (2006.01); C07D 521/00 (2006.01)

CPC (source: EP)

A61K 38/09 (2013.01); A61P 5/02 (2017.12); A61P 5/24 (2017.12); A61P 13/08 (2017.12); A61P 15/00 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 231/12 (2013.01); C07D 233/56 (2013.01); C07D 249/08 (2013.01); C07D 401/12 (2013.01); C07D 403/12 (2013.01); C07D 413/12 (2013.01); C07D 471/08 (2013.01); C07D 487/08 (2013.01)

Citation (search report)

  • No further relevant documents disclosed
  • See references of WO 9855119A1

Designated contracting state (EPC)

AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

DOCDB simple family (publication)

WO 9855119 A1 19981210; AU 7806998 A 19981221; CA 2291829 A1 19981210; EP 1011667 A1 20000628; EP 1011667 A4 20010328; JP 2002503252 A 20020129

DOCDB simple family (application)

US 9811204 W 19980601; AU 7806998 A 19980601; CA 2291829 A 19980601; EP 98926171 A 19980601; JP 50271499 A 19980601